SCHEMBL28828689

SCHEMBL28828689

CCOc1cccc(-c2cc3c(cc2OC)C(OC(N)=O)C(C)(C)C3)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
PDE7A Q13946 1/20 0.36
PDE3A Q14432 1/20 0.36
PDE10A Q9Y233 1/20 0.36
PTGS2 P35354 1/20 0.36
CD274 Q9NZQ7 2/20 0.35
HSD17B10 Q99714 1/20 0.35
PDCD1 Q15116 1/20 0.35
GRM5 P41594 1/20 0.35
GRM1 Q13255 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
ICMT O60725 2/20 0.35
DHODH Q02127 1/20 0.34
CHRM3 P20309 1/20 0.34
POLB P06746 1/20 0.34
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
SYK P43405 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828636 0.93 ERN1 (0.41) CD274GAAMAPTDHODHPRMT5
SCHEMBL28828396 0.92 NR1H4 (0.37) DHODHCHRM3
SCHEMBL28828506 0.91 CYP1A1 (0.40) HSD17B10GAAMAPTDHODHSYK
SCHEMBL28828597 0.90 PRMT5 (0.37) DHODHPRMT5WDR77
SCHEMBL28828389 0.89 ALDH1A1 (0.37) HSD17B10GAAMAPTMAPK1
SCHEMBL28828664 0.88 PTGS2 (0.45) RXRARXRBPTGS2GAAMAPT
SCHEMBL29121368 0.88 PTGS2 (0.45) RXRARXRBPTGS2GAAMAPT
SCHEMBL28828663 0.88 RXRA (0.36) RXRARXRBMAPTDHODH
SCHEMBL28828531 0.87 LMNA (0.36)
SCHEMBL28828550 0.85 RXRA (0.47) RXRARXRBGAAMAPTICMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed