SCHEMBL28828451

SCHEMBL28828451

COc1cc2c(cc1-c1cccc(C(C)C)c1)CC(C)(C)C2OC(N)=O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSA P10619 9/20 0.38
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
HDAC4 P56524 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
MTNR1B P49286 1/20 0.33
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828393 0.90 AKR1C3 (0.37) CTSAAKR1C3AKR1C2
SCHEMBL28828663 0.88 RXRA (0.36) AKR1C3AKR1C2RXRARXRB
SCHEMBL28828506 0.88 CYP1A1 (0.40) HDAC4HDAC8
SCHEMBL28828464 0.87 F2R (0.39) CTSA
SCHEMBL29121190 0.87 RXRA (0.34) AKR1C3AKR1C2RXRARXRBRXRG
SCHEMBL28828502 0.87 RXRA (0.34) AKR1C3AKR1C2RXRARXRBRXRG
SCHEMBL28828535 0.87 HTR7 (0.34) CTSAAKR1C3AKR1C2MTNR1B
SCHEMBL28828446 0.86 OTUD7B (0.43) CTSAAKR1C3AKR1C2
SCHEMBL28828501 0.84 RXRA (0.44) HDAC4HDAC8RXRARXRBRXRG
SCHEMBL29121307 0.84 RXRA (0.44) HDAC4HDAC8RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed