SCHEMBL28828684

SCHEMBL28828684

CC1(C)Cc2ccc(-c3ccc(C(F)(F)F)cc3)cc2C1OC(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 8/20 0.43
TDP2 O95551 1/20 0.38
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
DHODH Q02127 1/20 0.36
HDAC2 Q92769 2/20 0.36
SIGMAR1 Q99720 1/20 0.35
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
KCNH2 Q12809 1/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828662 0.91 KIF11 (0.43) KIF11TDP2CYP11B1CYP11B2DHODH
SCHEMBL28828505 0.90 KIF11 (0.44) KIF11
SCHEMBL29228304 0.89 KIF11 (0.41) KIF11TDP2CYP11B1CYP11B2DHODH
SCHEMBL28950173 0.87 KLKB1 (0.36) HDAC2HDAC1
SCHEMBL28828515 0.86 PPIB (0.40) KIF11DHODH
SCHEMBL28828381 0.85 KIF11 (0.34) KIF11DHODH
SCHEMBL28828623 0.84 JAK2 (0.35) TDP2HDAC2BRD4BRD2BRD3
SCHEMBL28828657 0.83 PGR (0.34)
SCHEMBL28828437 0.83 PGR (0.34) CYP11B1CYP11B2HDAC2PSEN1PSEN2
SCHEMBL28828548 0.83 KDM4E (0.38) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed