SCHEMBL28829583

SCHEMBL28829583

COc1cccc(I)c1NOC(=O)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
ELANE P08246 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
ALOX12 P18054 1/20 0.36
GAA P10253 1/20 0.35
MAPT P10636 3/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
ATM Q13315 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28829531 0.81 CYP3A4 (0.41) LMNAGAAMAPTSMN1; SMN2MEN1
SCHEMBL14042913 0.79 KDM4E (0.50) CA12CA1CA2CA7CA9
SCHEMBL28018573 0.75 KDM4E (0.52) KDM4ELMNAALOX12GAAMAPT
SCHEMBL729159 0.73 ATR (0.42) CA12CA1CA2CA7CA9
SCHEMBL28060869 0.73 PDK1 (0.43) CA12CA1CA2CA7CA9
SCHEMBL5361399 0.73 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL24926410 0.67 ELANE (0.53) CA12CA1CA2CA7CA9
SCHEMBL28370638 0.67 ELANE (0.62) ELANELMNAMAPTNPSR1
SCHEMBL364665 0.67 ELANE (0.53) ELANELMNAMAPTNPSR1ALDH1A1
SCHEMBL31031255 0.67 ELANE (0.53) ELANELMNAMAPTNPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103214482-B Imidazo [1,2-a] pyridine compounds as receptor tyrosine kinase inhibitors 阵列生物制药公司 2016-06-29 CN disclosed