SCHEMBL2882981

SCHEMBL2882981

CN1CCC(c2ccccc2)C(CO)C1

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 3/20 0.54
SLC6A2 P23975 2/20 0.54
SLC6A4 P31645 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5459465 1.00 SLC6A3 (0.54) SLC6A3SLC6A2SLC6A4
SCHEMBL4759736 1.00 SLC6A3 (0.54) SLC6A3SLC6A2SLC6A4
SCHEMBL4759732 1.00 SLC6A3 (0.54) SLC6A3SLC6A2SLC6A4
SCHEMBL5459468 1.00 SLC6A3 (0.54) SLC6A3SLC6A2SLC6A4
SCHEMBL6826523 0.86 SLC6A3 (0.54) SLC6A3
SCHEMBL3436817 0.85 MEN1 (0.46) SLC6A3SLC6A2SLC6A4
SCHEMBL3832793 0.84 SLC6A3 (0.72) SLC6A3
SCHEMBL3833873 0.84 SLC6A3 (0.72) SLC6A3
SCHEMBL1944023 0.84 SLC6A3 (0.52) SLC6A3
SCHEMBL7812342 0.84 SLC6A3 (0.72) SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015071831-A1 AN IMPROVED PROCESS FOR MINIMISING THE FORMATION OF DEHALOGENATED BYPRODUCTS Piramal Enterprises Limited (IN) 2015-05-21 WO disclosed
US-7855294-B2 Cycloalkanopyridine derivative BANYU PHARMACEUTICAL CO., LTD. (JP) 2010-12-21 US disclosed
EP-1966137-A2 PIPERIDINE DERIVATIVES Pfizer Products Inc. (US) 2008-09-10 EP disclosed
US-20070191419-A1 Cycloalkanopyridine derivative MSD K.K. (JP) 2007-08-16 US disclosed
WO-2007072150-A2 PIPERIDINE DERIVATIVES PFIZER PRODUCTS INC. (US) 2007-06-28 WO disclosed
US-20070142389-A1 PIPERIDINE DERIVATIVES PFIZER INC. (US) 2007-06-21 US disclosed
US-20070142389-A1 PIPERIDINE DERIVATIVES PFIZER INC. (US) 2007-06-21 US disclosed
WO-2007034270-A2 IMPROVED PROCESS FOR THE PREPARATION OF (-) TRANS-N-METHYL PAROXETINE ORCHID CHEMICALS & PHARMACEUTICALS LIMITED (IN) 2007-03-29 WO disclosed
EP-1726590-A1 CYCLOALKANOPYRIDINE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2006-11-29 EP disclosed
WO-2004043921-A1 NOVEL PROCESS FOR THE PREPARATION OF 4-ARYL-3-HYDROXYMETHYL-1-METHYLPIPERIDINES. NATCO PHARMA LIMITED (IN) 2004-05-27 WO disclosed
CN-1068597-C Process for preparing 4 -aryl -piperidine derivatives NOVO NORDISK AS (DK) 2001-07-18 CN disclosed
EP-1074550-A1 Process for the preparation of 3-substituted 4-phenyl-piperidine derivatives CHEMI S.p.A. (IT) 2001-02-07 EP disclosed
WO-2000020390-A1 MONOMERIC AND DIMERIC HETEROCYCLES, AND THERAPEUTIC USES THEREOF GEORGETOWN UNIVERSITY (US) 2000-04-13 WO disclosed
CN-1184476-A Process for preparing 4 -aryl -piperidine derivatives NOVO NORDISK AS (DK) 1998-06-10 CN disclosed
EP-0828735-A1 PROCESS FOR PREPARING 4-ARYL-PIPERIDINE DERIVATIVES NOVO NORDISK A/S (DK) 1998-03-18 EP disclosed
WO-1996036636-A1 PROCESS FOR PREPARING 4-ARYL-PIPERIDINE DERIVATIVES NOVO NORDISK A/S (DK) 1996-11-21 WO disclosed
EP-0284395-B1 NOVEL GLYCEROL DERIVATIVE AND ANTI-HYPERTENSIVE AGENT NIPPON CHEMIPHAR CO., LTD. (JP) 1993-06-23 EP disclosed
US-5183811-A Glycerol derivative and anti-hypertensive agent NIPPON CHEMIPHAR CO., LTD. (JP) 1993-02-02 US disclosed
US-4962096-A WITH REDUCED PLATELET AGGREGATING ACTION NIPPON CHEMIPHAR CO., LTD. (JP) 1990-10-09 US disclosed
EP-0284395-A2 Novel glycerol derivative and anti-hypertensive agent NIPPON CHEMIPHAR CO., LTD. (JP) 1988-09-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070142389-A1 PIPERIDINE DERIVATIVES CFTR, HDAC10, RPP30 SLC6A3 2127/4885SLC6A2 2730/4885SLC6A4 1044/4885
US-20070191419-A1 Cycloalkanopyridine derivative OPRL1, OPRK1, AVPR2 SLC6A3 58/4885SLC6A2 150/4885SLC6A4 241/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.