SCHEMBL28830147

SCHEMBL28830147

CNc1cc(N2CCC(C(F)(F)F)CC2)c(C(F)(F)F)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.40
PIK3R1 P27986 1/20 0.39
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CCNA1 P78396 1/20 0.36
AR P10275 1/20 0.36
PROKR1 Q8TCW9 3/20 0.35
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
SCN10A Q9Y5Y9 2/20 0.33
TRPV1 Q8NER1 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
EPHX2 P34913 4/20 0.33
CYP2C9 P11712 2/20 0.33
LRRK2 Q5S007 1/20 0.33
WNT1 P04628 1/20 0.32
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16635418 0.80 TRPA1 (0.42) TRPA1PIK3R1CCNA2CDK2CCNA1
SCHEMBL16635362 0.76 TRPA1 (0.46) TRPA1ARKDM4EMAPTSCN10A
SCHEMBL16635293 0.76 AR (0.43) TRPA1ARKDM4ECYP3A4
Hydrochloric Acid SCHEMBL17959625 0.75 TRPA1 (0.45) TRPA1ARKDM4EMAPTSCN10A
SCHEMBL28017904 0.74 HRH4 (0.43) TRPA1KDM4EMAPT
SCHEMBL28864068 0.71 CYP46A1 (0.40) TRPA1KDM4EMAPTCYP1A2CYP3A4
SCHEMBL9900024 0.70 SCN10A (0.35) TRPA1KDM4EMAPTCYP1A2CYP3A4
SCHEMBL15033706 0.69 AR (0.34) TRPA1ARKDM4EMAPTSCN10A
SCHEMBL30834536 0.67 NNMT (0.46) PIK3R1CYP1A2CYP3A4LRRK2
SCHEMBL11916195 0.67 CYP1A2 (0.44) PIK3R1CYP1A2CYP3A4LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105612153-A Substituted sulfonamide compounds as TRPA1 conditioner HOFFMANN LA ROCHE 2016-05-25 CN disclosed