SCHEMBL28832015

SCHEMBL28832015

COc1cccc2ccc(=O)n(CC(=O)ONC(=O)c3ccc(C(C)(C)C)cc3)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
LMNA P02545 4/20 0.38
KDM4E B2RXH2 2/20 0.38
KMT2A Q03164 6/20 0.37
MEN1 O00255 5/20 0.37
MAPT P10636 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
HTR6 P50406 1/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 2/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
ALOX15 P16050 1/20 0.36
APEX1 P27695 1/20 0.36
MAPK1 P28482 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28831998 0.91 SMN1; SMN2 (0.41) ALDH1A1KDM4EKMT2AMAPTDRD2
SCHEMBL29143300 0.78 HTR6 (0.44) ALDH1A1LMNAKDM4EKMT2AMEN1
SCHEMBL11999976 0.75 MEN1 (0.52) ALDH1A1LMNAKDM4EKMT2AMEN1
SCHEMBL5040066 0.74 HTR6 (0.47) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL12002188 0.69 HTR6 (0.50) ALDH1A1KDM4EKMT2AMEN1HTR6
SCHEMBL2799840 0.68 HTR6 (0.47) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL28294733 0.67 HDAC1 (0.53) ALDH1A1LMNAKMT2AMEN1MAPT
SCHEMBL2797396 0.66 HTR6 (0.47) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL4225409 0.65 PTGER3 (0.49) ALDH1A1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL28832153 0.64 MAPT (0.46) ALDH1A1LMNAKDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114702444-A AHA1 inhibitor with multiple myeloma resisting effect and preparation method and application thereof 南京中医药大学 2022-07-05 CN disclosed