SCHEMBL28831998

SCHEMBL28831998

COc1cccc2ccc(=O)n(CC(=O)ONC(=O)c3ccc(F)cc3)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.41
HTR6 P50406 1/20 0.39
ALDH1A1 P00352 4/20 0.38
HPGD P15428 2/20 0.38
HTR1A P08908 4/20 0.37
DRD2 P14416 2/20 0.37
KMT2A Q03164 2/20 0.37
CACNA1B Q00975 1/20 0.37
APBA1 Q02410 1/20 0.37
KDM4E B2RXH2 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CXCR3 P49682 1/20 0.36
DRD4 P21917 1/20 0.36
ADRA1D P25100 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28832015 0.91 ALDH1A1 (0.38) SMN1; SMN2RAB9AHTR6ALDH1A1DRD2
SCHEMBL29143300 0.81 HTR6 (0.44) SMN1; SMN2GAAHTR6ALDH1A1KMT2A
SCHEMBL11999976 0.77 MEN1 (0.52) GAARAB9AHTR6ALDH1A1KMT2A
SCHEMBL5040066 0.76 HTR6 (0.47) SMN1; SMN2GAAHTR6ALDH1A1HPGD
SCHEMBL12002188 0.71 HTR6 (0.50) GAAHTR6ALDH1A1KMT2AKDM4E
SCHEMBL2799840 0.70 HTR6 (0.47) GAAHTR6ALDH1A1HPGDKMT2A
SCHEMBL28262932 0.68 ALDH1A1 (0.47) SMN1; SMN2GAARAB9AALDH1A1HPGD
SCHEMBL2797396 0.68 HTR6 (0.47) SMN1; SMN2GAARAB9AHTR6ALDH1A1
SCHEMBL4225409 0.67 PTGER3 (0.49) SMN1; SMN2ALDH1A1KMT2AKDM4EHSD17B10
SCHEMBL98218 0.65 CYP19A1 (0.54) SMN1; SMN2GAARAB9AHTR6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114702444-A AHA1 inhibitor with multiple myeloma resisting effect and preparation method and application thereof 南京中医药大学 2022-07-05 CN disclosed