SCHEMBL29143300

SCHEMBL29143300

COc1cccc2ccc(=O)n(CC(=O)ON)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.44
CCR2 P41597 1/20 0.39
KDM4E B2RXH2 5/20 0.39
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37
CCND2 P30279 1/20 0.37
CCND3 P30281 1/20 0.37
MAPT P10636 4/20 0.36
ALDH1A1 P00352 3/20 0.36
KMT2A Q03164 4/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
MEN1 O00255 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
GAA P10253 3/20 0.36
MAPK1 P28482 1/20 0.36
CYP19A1 P11511 1/20 0.36
NQO2 P16083 1/20 0.36
CYP2A6 P11509 1/20 0.35
POLB P06746 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11999976 0.86 MEN1 (0.52) HTR6KDM4EMAPTALDH1A1KMT2A
SCHEMBL5040066 0.85 HTR6 (0.47) HTR6CCR2KDM4EMAPTALDH1A1
SCHEMBL28831998 0.81 SMN1; SMN2 (0.41) HTR6KDM4EMAPTALDH1A1KMT2A
SCHEMBL12002188 0.79 HTR6 (0.50) HTR6CCR2KDM4ECDK4CCND1
SCHEMBL28832015 0.78 ALDH1A1 (0.38) HTR6KDM4EMAPTALDH1A1KMT2A
SCHEMBL2799840 0.78 HTR6 (0.47) HTR6CCR2KDM4EMAPTALDH1A1
SCHEMBL2797396 0.75 HTR6 (0.47) HTR6CCR2KDM4EMAPTALDH1A1
SCHEMBL98218 0.72 CYP19A1 (0.54) HTR6KDM4EMAPTALDH1A1KMT2A
SCHEMBL4225409 0.72 PTGER3 (0.49) KDM4ECDK4CCND1CCND2CCND3
SCHEMBL2800552 0.68 HTR6 (0.39) HTR6CCR2KDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117186001-A AHA1 inhibitor with multiple myeloma-resisting activity and preparation method and application thereof 南京中医药大学 2023-12-08 CN disclosed
CN-114702444-B AHA1 inhibitor with multiple myeloma resistance and preparation method and application thereof 南京中医药大学 2023-09-12 CN disclosed