SCHEMBL28833548

SCHEMBL28833548

COc1cc(-c2nc(-c3ccc(F)cc3)n[nH]2)cc(OC)c1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.57
POLB P06746 1/20 0.57
TSHR P16473 1/20 0.57
PSEN1 P49768 1/20 0.57
PSEN2 P49810 1/20 0.57
APH1B Q8WW43 1/20 0.57
NCSTN Q92542 1/20 0.57
APH1A Q96BI3 1/20 0.57
PSENEN Q9NZ42 1/20 0.57
GRK6 P43250 1/20 0.46
FYN P06241 1/20 0.46
HSD17B10 Q99714 2/20 0.46
MAP3K11 Q16584 2/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 1/20 0.44
MPI P34949 1/20 0.44
APOBEC3G Q9HC16 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
NR1H2 P55055 2/20 0.44
NR1H3 Q13133 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28075488 0.87 KDM4E (0.58) KDM4EPOLBTSHRGRK6FYN
SCHEMBL28096008 0.86 KDM4E (0.55) KDM4EPOLBTSHRPSEN1PSEN2
SCHEMBL28095606 0.86 KDM4E (0.55) KDM4EPOLBTSHRPSEN1PSEN2
SCHEMBL28095619 0.86 KDM4E (0.57) KDM4EPOLBTSHRPSEN1PSEN2
SCHEMBL17279690 0.86 NR1H2 (0.60) KDM4EPOLBTSHRGRK6ALDH1A1
SCHEMBL28096011 0.84 KDM4E (0.55) KDM4EPOLBTSHRPSEN1PSEN2
SCHEMBL15026741 0.83 PSEN1 (0.63) KDM4EPSEN1PSEN2APH1BNCSTN
SCHEMBL17280055 0.83 KDM4E (0.60) KDM4EPOLBTSHRPSEN1PSEN2
SCHEMBL28075481 0.83 KDM4E (0.57) KDM4EPOLBTSHRPSEN1PSEN2
SCHEMBL28096010 0.81 KDM4E (0.55) KDM4EPOLBTSHRGRK6HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106243130-B 3,6- diaryl-[1,2,4] triazole simultaneously [3,4-b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2019-03-01 CN claimed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN claimed
CN-106243130-B 3,6- diaryl-[1,2,4] triazole simultaneously [3,4-b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2019-03-01 CN disclosed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN disclosed