SCHEMBL28833892

SCHEMBL28833892

CC(C)c1cccc(C(c2ccccc2)(c2ccccc2)N2C[C@@H]2C(=O)OCc2ccccc2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 7/20 0.39
CTSL P07711 1/20 0.38
HTR2C P28335 1/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
HPGD P15428 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
BCL9 O00512 2/20 0.36
CTNNB1 P35222 2/20 0.36
GLRA1 P23415 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362332 0.86 FKBP1A (0.45) FKBP1AHTR2CHPGDALDH1A1TSHR
SCHEMBL9367912 0.86 FKBP1A (0.45) FKBP1AHTR2CHPGDALDH1A1TSHR
SCHEMBL28833932 0.83 NOTUM (0.44) HPGDALDH1A1CYP3A4SLC6A9
SCHEMBL28838606 0.77 ALDH1A1 (0.45) ALDH1A1POLBACE
SCHEMBL7122146 0.76 POLB (0.43) FKBP1AHTR2CHPGDALDH1A1POLB
SCHEMBL28975603 0.74 FKBP1A (0.49) FKBP1AHTR2CCYP2C19TSHR
SCHEMBL28975604 0.74 FKBP1A (0.49) FKBP1AHTR2CCYP2C19TSHR
SCHEMBL7125855 0.73 FKBP1A (0.40) FKBP1AHTR2CHPGDALDH1A1TSHR
SCHEMBL7247064 0.73 FKBP1A (0.40) FKBP1AHTR2CHPGDALDH1A1TSHR
SCHEMBL28838626 0.73 S1PR1 (0.40) CHRM3ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114980976-A Covalent RAS inhibitors and uses thereof 锐新医药公司 2022-08-30 CN disclosed
CN-114901366-A RAS inhibitors 锐新医药公司 2022-08-12 CN disclosed