SCHEMBL288347

SCHEMBL288347

Cc1ccc(NS(=O)(=O)n2ccnc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 1/20 0.49
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
TSHR P16473 1/20 0.45
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HPGD P15428 3/20 0.43
HTT P42858 2/20 0.43
ALDH1A1 P00352 4/20 0.42
TP53 P04637 1/20 0.42
CYP19A1 P11511 2/20 0.41
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
LMNA P02545 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14080961 0.85 KMT2A (0.42) CA1CA2TSHRKMT2AMEN1
SCHEMBL27855435 0.76 TSHR (0.46) TSHRKMT2AMEN1HPGDHTT
SCHEMBL217862 0.76 TP53 (0.69) CA1CA2TSHRKMT2AMEN1
Ammonia Solution, Strong SCHEMBL28097128 0.75 TP53 (0.67) CA1CA2TSHRKMT2AMEN1
SCHEMBL12765340 0.72 HTT (0.53) TSHRKMT2AMEN1SMN1; SMN2L3MBTL1
SCHEMBL13236227 0.72 HTT (0.52) TSHRKMT2AMEN1SMN1; SMN2L3MBTL1
Toluene SCHEMBL28953742 0.70 TSHR (0.45) TSHRKMT2AMEN1SMN1; SMN2L3MBTL1
SCHEMBL31191242 0.69 HTT (0.50) TSHRKMT2AMEN1SMN1; SMN2L3MBTL1
SCHEMBL16720612 0.68 ALDH1A1 (0.43) KMT2AMEN1SMN1; SMN2L3MBTL1HPGD
SCHEMBL27062690 0.68 HTT (0.48) TSHRKMT2AMEN1SMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 72 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922831-A1 PESTICIDAL COMPOUNDS BASED ON ARYLTHIOSULFONAMIDE DERIVATIVES Syngenta Participations AG (CH) 2015-09-30 EP disclosed
EP-2922837-A1 INSECTICIDAL COMPOUNDS BASED ON N-(ARYLSULFANYLMETHYL) CARBOXAMIDE DERIVATIVES Syngenta Participations AG (CH) 2015-09-30 EP disclosed
EP-2917201-A1 DIHYDROTHIOPHENE DERIVATIVES AS INSECTICIDAL COMPOUNDS Syngenta Participations AG (CH) 2015-09-16 EP disclosed
EP-2887810-A1 METHODS OF CONTROLLING INSECTS Syngenta Participations AG (CH) 2015-07-01 EP disclosed
EP-2887802-A2 METHODS OF SOIL PEST CONTROL Syngenta Participations AG (CH) 2015-07-01 EP disclosed
EP-2887809-A1 METHODS OF CONTROLLING INSECTS Syngenta Participations AG (CH) 2015-07-01 EP disclosed
WO-2014079935-A9 INSECTICIDAL COMPOUNDS BASED ON ARYLTHIOACETAMIDE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2014-09-04 WO disclosed
EP-2748154-A1 PROCESS FOR THE PREPARATION OF THIETANE DERIVATIVES Syngenta Participations AG (CH) 2014-07-02 EP disclosed
EP-2748155-A1 ISOXAZOLINE DERIVATIVES AS INSECTICIDAL COMPOUNDS Syngenta Participations AG (CH) 2014-07-02 EP disclosed
EP-2748137-A1 DIHYDROFURAN DERIVATIVES AS INSECTICIDAL COMPOUNDS Syngenta Participations AG (CH) 2014-07-02 EP disclosed
WO-2011067240-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067135-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067203-A1 CHEMICAL COMPOUNDS AND THEIR USE AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067131-A1 SPIROHETEROCYCLIC DIONE DERIVATIVES USED AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067272-A1 INSECTICIDAL COMPOUNDS BASED ON ISOXAZOLINE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
EP-2324010-A1 INSECTICIDAL PHENYL- OR PYRIDYL-PIPERIDINE COMPOUNDS Syngenta Participations AG (CH) 2011-05-25 EP disclosed
WO-2011003684-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2011-01-13 WO disclosed
WO-2010066780-A1 SPIROHETEROCYCLIC N-OXYPIPERIDINES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-06-17 WO disclosed
WO-2010063670-A1 SPIROHETEROCYCLIC N-OXYAMIDES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-06-10 WO disclosed
WO-2001055140-A1 ISOTHIAZOLE DERIVATIVES AND THEIR USE AS PESTICIDES SYNGENTA LIMITED (GB) 2001-08-02 WO disclosed