SCHEMBL28839743

SCHEMBL28839743

Brc1ncnc2[nH]ncc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.63
RET P07949 1/20 0.63
PI4KA P42356 1/20 0.63
LRRK2 Q5S007 1/20 0.63
PI4K2B Q8TCG2 1/20 0.63
PI4K2A Q9BTU6 1/20 0.63
PI4KB Q9UBF8 1/20 0.63
PDPK1 O15530 1/20 0.57
CHEK1 O14757 1/20 0.55
AURKA O14965 1/20 0.55
MKNK1 Q9BUB5 3/20 0.54
MAPK1 P28482 2/20 0.54
ALDH1A1 P00352 1/20 0.49
HPGDS O60760 1/20 0.49
CYP1A2 P05177 2/20 0.46
CCNT1 O60563 1/20 0.46
CCNA2 P20248 1/20 0.46
CDK2 P24941 1/20 0.46
CDK9 P50750 1/20 0.46
CCNA1 P78396 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30763272 1.00 XDH (0.63) XDHRETPI4KALRRK2PI4K2B
SCHEMBL11363 0.77 XDH (1.00) XDHRETPI4KALRRK2PI4K2B
SCHEMBL29351045 0.77 XDH (1.00) XDHRETPI4KALRRK2PI4K2B
Tisopurine SCHEMBL93974 0.76 XDH (0.61) XDHRETPI4KALRRK2PI4K2B
SCHEMBL11218 0.76 XDH (0.61) XDHRETPI4KALRRK2PI4K2B
SCHEMBL2619226 0.76 RET (0.61) XDHRETPI4KALRRK2PI4K2B
SCHEMBL15504523 0.76 XDH (0.61) XDHRETPI4KALRRK2PI4K2B
Hydrochloric Acid SCHEMBL14742346 0.76 XDH (0.96) XDHRETPI4KALRRK2PI4K2B
SCHEMBL4975495 0.76 XDH (0.61) XDHRETPI4KALRRK2PI4K2B
Allopurinol SCHEMBL4627 0.76 XDH (0.61) XDHRETPI4KALRRK2PI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117586267-A Preparation method of 4-bromopyrazole [3,4-D ] -pyrimidine 山东百启生物医药有限公司 2024-02-23 CN claimed
CN-115043841-B Preparation and application of heterocyclic compound serving as BTK inhibitor 药雅科技(上海)有限公司 2024-04-09 CN disclosed
CN-117586267-A Preparation method of 4-bromopyrazole [3,4-D ] -pyrimidine 山东百启生物医药有限公司 2024-02-23 CN disclosed
CN-117586267-A Preparation method of 4-bromopyrazole [3,4-D ] -pyrimidine 山东百启生物医药有限公司 2024-02-23 CN disclosed
CN-115043832-B FGFR inhibitor acetylenic heterocyclic compound and preparation method and application thereof 药雅科技(上海)有限公司 2023-08-22 CN disclosed
CN-115043841-A Preparation and application of heterocyclic compound as BTK inhibitor 药雅科技(上海)有限公司 2022-09-13 CN disclosed
CN-115043832-A FGFR inhibitor alkyne-substituted heterocyclic compound and preparation method and application thereof 药雅科技(上海)有限公司 2022-09-13 CN disclosed