SCHEMBL28840767

SCHEMBL28840767

N#CCc1ccc2c(c1)COCC2

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 2/20 0.38
WDR77 Q9BQA1 2/20 0.38
ROCK2 O75116 1/20 0.34
ENPP2 Q13822 1/20 0.33
MMP3 P08254 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
KIF11 P52732 1/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PIK3CD O00329 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27582186 0.86 ENPP2 (0.37) ENPP2MMP3KDM4ETDP1KIF11
SCHEMBL29790934 0.86 ENPP2 (0.37) ENPP2MMP3KDM4ETDP1KIF11
SCHEMBL4521078 0.78 ENPP2 (0.39) ENPP2MMP3KDM4ETDP1TSHR
SCHEMBL21382504 0.77 PRMT5 (0.38) PRMT5WDR77PIK3CD
SCHEMBL28840799 0.77 PRMT5 (0.38) PRMT5WDR77PIK3CD
SCHEMBL21382554 0.77 PRMT5 (0.40) PRMT5WDR77PIK3CD
SCHEMBL9123053 0.77 PRMT5 (0.38) PRMT5WDR77KDM4ENPC1RAB9A
SCHEMBL1466419 0.77 RXRB (0.40) ENPP2MMP3KDM4ETDP1NPC1
SCHEMBL8089040 0.75 RAB9A (0.44) NPC1RAB9A
SCHEMBL3642604 0.75 CHRM2 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114907389-A Boronic acid derivatives 首药控股(北京)股份有限公司 2022-08-16 CN disclosed