SCHEMBL28840783

SCHEMBL28840783

O=C1CCCn2c1c(C(I)C(=O)O)c1ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.40
CREBBP Q92793 1/20 0.40
MTNR1A P48039 6/20 0.38
MTNR1B P49286 6/20 0.38
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 4/20 0.38
CYP1A2 P05177 2/20 0.38
HSD17B10 Q99714 2/20 0.38
USP2 O75604 1/20 0.38
BCHE P06276 1/20 0.38
CFTR P13569 1/20 0.38
ALOX15 P16050 1/20 0.38
ACHE P22303 1/20 0.38
HKDC1 Q2TB90 1/20 0.38
GOPC Q9HD26 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PABPC1 P11940 1/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28922903 0.81 KDM4E (0.35) TP53CREBBPKDM4EALDH1A1CYP1A2
SCHEMBL28840719 0.74 TERT (0.47) TP53CREBBPMTNR1AMTNR1BKDM4E
SCHEMBL16201684 0.72 CDK5 (0.45) TP53CREBBPMTNR1AMTNR1BKDM4E
SCHEMBL10725922 0.72 KDM4E (0.54) TP53CREBBPMTNR1AMTNR1BKDM4E
SCHEMBL9471252 0.71 MTNR1A (0.46) TP53CREBBPMTNR1AMTNR1BKDM4E
SCHEMBL7384938 0.67 MTNR1A (0.41) TP53CREBBPMTNR1AMTNR1BKDM4E
SCHEMBL18202181 0.65 PABPC1 (0.49) TP53CREBBPMTNR1AMTNR1BKDM4E
SCHEMBL7321799 0.63 HTR2A (0.52) KDM4EALDH1A1HSD17B10ALOX15MEN1
SCHEMBL31486786 0.63 HTR2A (0.52) KDM4EALDH1A1HSD17B10ALOX15MEN1
SCHEMBL16201678 0.63 PABPC1 (0.46) TP53CREBBPMTNR1AMTNR1BPABPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114907389-A Boronic acid derivatives 首药控股(北京)股份有限公司 2022-08-16 CN disclosed