SCHEMBL28840935

SCHEMBL28840935

COc1cc(O)c2c(c1OC)OC(c1ccccc1)C(=O)C2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.46
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
PABPC1 P11940 1/20 0.41
APEX1 P27695 1/20 0.41
RECQL P46063 1/20 0.41
KMT2A Q03164 1/20 0.41
EIF4H Q15056 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ACHE P22303 1/20 0.40
PLK1 P53350 1/20 0.40
BACE1 P56817 1/20 0.40
SIRT1 Q96EB6 2/20 0.38
ABCG2 Q9UNQ0 3/20 0.38
ABCB1 P08183 2/20 0.38
TUBB4A P04350 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28513252 0.91 CYP19A1 (0.46) CYP19A1MEN1POLBGAAMAPT
SCHEMBL17503283 0.90 NPC1 (0.45) CYP19A1MEN1POLBGAAMAPT
SCHEMBL17907267 0.89 KMT2A (0.50) CYP19A1MEN1POLBGAAMAPT
SCHEMBL28879340 0.89 ABCG2 (0.42) CYP19A1MEN1POLBGAAMAPT
SCHEMBL2124063 0.87 TUBB4A (0.47) CYP19A1MAPTNPC1RAB9AABCG2
SCHEMBL665266 0.83 CYP19A1 (0.51) CYP19A1MEN1POLBGAAMAPT
SCHEMBL29204371 0.81 CYP19A1 (0.42) CYP19A1MEN1POLBGAAMAPT
SCHEMBL17907271 0.81 KMT2A (0.44) CYP19A1MEN1POLBGAAMAPT
SCHEMBL27950799 0.81 TAS2R31 (0.39) CYP19A1MEN1POLBMAPTKMT2A
SCHEMBL10425234 0.79 KDM4E (0.46) NPC1RAB9ASIRT1ABCG2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115068491-A Medical application of andrographolide as LTB4 receptor inhibitor 中国医学科学院药物研究所 2022-09-20 CN disclosed
CN-115068467-A Medical application of andrographolide as LTB4 receptor inhibitor 中国医学科学院药物研究所 2022-09-20 CN disclosed