SCHEMBL28840974

SCHEMBL28840974

CCC(=O)c1cc(C(F)(F)F)c(Cl)cc1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 2/20 0.39
BRAF P15056 2/20 0.36
HDAC1 Q13547 2/20 0.36
KDR P35968 1/20 0.36
DDR1 Q08345 1/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NOTUM Q6P988 2/20 0.35
KCNJ5 P48544 1/20 0.35
KCNJ3 P48549 1/20 0.35
P2RX7 Q99572 1/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
HDAC3 O15379 1/20 0.34
RAF1 P04049 1/20 0.34
ARAF P10398 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16637275 0.82 CFTR (0.42) CFTRBRAFHDAC1KDRALDH1A1
SCHEMBL9559940 0.81 CYP3A4 (0.41) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL16528370 0.81 KDM4E (0.46) CFTRALDH1A1KDM4EHSD17B10MAPT
SCHEMBL16528992 0.80 ALDH1A1 (0.50) CFTRKDRALDH1A1KDM4EHPGD
SCHEMBL16637057 0.78 CFTR (0.64) CFTRKDRALDH1A1KDM4EHPGD
SCHEMBL23040875 0.76 CFTR (0.45) CFTRBRAFHDAC1KDRALDH1A1
SCHEMBL29417318 0.76 CFTR (0.45) CFTRBRAFHDAC1KDRALDH1A1
SCHEMBL19554287 0.75 CFTR (0.49) CFTRALDH1A1KDM4EHSD17B10MAPT
SCHEMBL3549347 0.73 CFTR (0.51) CFTRKDRALDH1A1KDM4EHPGD
SCHEMBL25223342 0.72 SLC9A1 (0.37) ALDH1A1KDM4EHPGDLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106488910-A Inhibitors of kras g12c 亚瑞克西斯制药公司 2017-03-08 CN disclosed