SCHEMBL28841998

SCHEMBL28841998

CN(C)/C=N/c1ccc(NC(=S)NC(C)(C)CNC(=O)OC(C)(C)C)cc1C#N

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
RORC P51449 4/20 0.33
AR P10275 2/20 0.33
PTPN11 Q06124 1/20 0.33
MAPKAPK2 P49137 5/20 0.33
AAK1 Q2M2I8 1/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
NSD2 O96028 1/20 0.31
POLB P06746 1/20 0.31
HTT P42858 1/20 0.31
TRPA1 O75762 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28842000 1.00 ALDH1A1 (0.37) ALDH1A1GAARORCARPTPN11
SCHEMBL22619977 0.89 POLB (0.35) ALDH1A1GAAARPOLBHTT
SCHEMBL20605383 0.89 POLB (0.35) ALDH1A1GAAARPOLBHTT
SCHEMBL28841996 0.85 MAPT (0.32) ALDH1A1ARPOLBHTT
SCHEMBL1192514 0.85 POLB (0.38) ALDH1A1GAAPOLBHTT
SCHEMBL20838797 0.85 POLB (0.38) ALDH1A1GAAPOLBHTT
SCHEMBL29677017 0.85 POLB (0.38) ALDH1A1GAAPOLBHTT
SCHEMBL1192515 0.85 POLB (0.38) ALDH1A1GAAPOLBHTT
SCHEMBL30125784 0.82 BCHE (0.40) ARPTPN11AAK1CA1CA2
SCHEMBL20605467 0.81 IDO1 (0.34) ALDH1A1GAAPOLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107141293-B Nitrogen-containing heterocyclic compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2022-09-23 CN disclosed
CN-115057861-A Nitrogen-containing heterocyclic compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2022-09-16 CN disclosed