SCHEMBL28843253

SCHEMBL28843253

O=CNC1=NCCc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.49
NOS2 P35228 1/20 0.49
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAOA P21397 2/20 0.41
CES1 P23141 1/20 0.38
MAOB P27338 2/20 0.35
CYP2A6 P11509 1/20 0.35
CYP19A1 P11511 5/20 0.33
PABPC1 P11940 1/20 0.33
PDPK1 O15530 1/20 0.33
PARP1 P09874 1/20 0.33
PARP10 Q53GL7 1/20 0.33
PARP11 Q9NR21 1/20 0.33
CYP11B2 P19099 3/20 0.33
MIF P14174 1/20 0.33
PKM P14618 1/20 0.33
MAPK1 P28482 1/20 0.33
MAPT P10636 1/20 0.33
CYP11B1 P15538 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572470 0.78 NOS3 (0.55) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL11745466 0.77 NOS3 (0.58) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL28328181 0.76 KMT2A (0.31) CES1CYP19A1
Hydrochloric Acid SCHEMBL11744315 0.75 NOS3 (0.56) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL5128271 0.74 NOS3 (0.55) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL21984859 0.72 KDM4E (0.54) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL27937579 0.72 NOS3 (0.45) NOS3NOS2ALDH1A1KDM4EMAOA
SCHEMBL25055314 0.69 NOS3 (0.45) NOS3NOS2ALDH1A1KDM4EMAOA
Hydrochloric Acid SCHEMBL9374659 0.69 GRIN2B (0.45) NOS3NOS2ALDH1A1KDM4EMAPT
SCHEMBL11749232 0.68 GAA (0.58) NOS3NOS2ALDH1A1KDM4EMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105228996-B Tetrahydroisoquinolines containing substituted azoles as factor XIa inhibitors 百时美施贵宝公司 2017-11-28 CN claimed
CN-106795118-B Heterocyclic compound and their purposes as relevant orphan receptor (ROR) the GAMMA-T inhibitor of retinoids 武田药品工业株式会社 2019-10-08 CN disclosed
CN-103987697-B Substituted tetrahydroisoquinoline compounds as factor XIA inhibitors 百时美施贵宝公司 2017-04-26 CN disclosed