SCHEMBL28844653

SCHEMBL28844653

CCOC(=O)c1cc2c(N)cc(Br)cc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.48
ALDH1A1 P00352 6/20 0.48
RAB9A P51151 5/20 0.48
HPGD P15428 4/20 0.48
NPC1 O15118 4/20 0.48
LMNA P02545 3/20 0.48
L3MBTL1 Q9Y468 3/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
HSD17B10 Q99714 1/20 0.48
MMP13 P45452 4/20 0.47
MMP2 P08253 3/20 0.47
MAPT P10636 6/20 0.47
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
GAA P10253 3/20 0.47
GLA P06280 1/20 0.47
ATM Q13315 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30995141 0.86 KDM4E (0.50) KDM4EALDH1A1RAB9AHPGDNPC1
SCHEMBL23148030 0.86 KDM4E (0.50) KDM4EALDH1A1RAB9AHPGDNPC1
SCHEMBL30995242 0.83 ALOX15 (0.52) KDM4EALDH1A1RAB9AHPGDNPC1
SCHEMBL31405949 0.83 KDM4E (0.48) KDM4EALDH1A1RAB9AHPGDNPC1
SCHEMBL4037610 0.83 KDM4E (0.48) KDM4EALDH1A1RAB9AHPGDNPC1
SCHEMBL30995243 0.83 ALOX15 (0.52) KDM4EALDH1A1RAB9AHPGDNPC1
SCHEMBL28844613 0.81 KDM4E (0.48) KDM4EALDH1A1RAB9AHPGDNPC1
SCHEMBL3622667 0.80 KDM4E (0.45) KDM4EALDH1A1RAB9AHPGDNPC1
SCHEMBL21772092 0.79 KDM4E (0.47) KDM4EALDH1A1RAB9AHPGDNPC1
SCHEMBL28844710 0.79 ALDH1A1 (0.44) KDM4EALDH1A1RAB9AHPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110483366-B Indole compound and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-09-16 CN disclosed