SCHEMBL28844677

SCHEMBL28844677

COc1ccc(-c2ccc(F)c3[nH]c(C(=O)O)cc23)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 8/20 0.54
TDO2 P48775 8/20 0.54
KDM4E B2RXH2 1/20 0.52
HPGD P15428 1/20 0.52
PTGS2 P35354 4/20 0.45
PTGS1 P23219 2/20 0.44
KMO O15229 2/20 0.42
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
PRKAB2 O43741 1/20 0.42
PRKAG1 P54619 1/20 0.42
PRKAA2 P54646 1/20 0.42
PRKAA1 Q13131 1/20 0.42
PRKAG3 Q9UGI9 1/20 0.42
PRKAG2 Q9UGJ0 1/20 0.42
PRKAB1 Q9Y478 1/20 0.42
EIF4A3 P38919 1/20 0.41
FBP1 P09467 1/20 0.40
HSD17B1 P14061 1/20 0.40
HSD17B2 P37059 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28844729 0.86 PRKCZ (0.43) IDO1TDO2PTGS2PTGS1
SCHEMBL1144985 0.81 KDM4E (0.77) IDO1TDO2KDM4EHPGDEIF4A3
SCHEMBL22394891 0.74 IDO1 (0.65) IDO1TDO2EIF4A3
SCHEMBL1144591 0.73 KDM4E (0.77) IDO1TDO2KDM4EHPGDEIF4A3
SCHEMBL1810986 0.72 RAB9A (0.51) PTGS2PTGS1KMOAKR1C3AKR1C2
SCHEMBL22747188 0.72 IDO1 (0.75) IDO1TDO2KDM4EHPGDEIF4A3
SCHEMBL29974758 0.72 IDO1 (0.75) IDO1TDO2KDM4EHPGDEIF4A3
SCHEMBL24113316 0.71 IDO1 (0.52) IDO1TDO2KDM4EHPGDEIF4A3
SCHEMBL24112536 0.71 KDM4E (0.60) IDO1TDO2KDM4EHPGDEIF4A3
SCHEMBL31652065 0.71 IDO1 (0.50) IDO1TDO2KDM4EHPGDAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110483366-B Indole compound and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-09-16 CN disclosed