SCHEMBL28844931

SCHEMBL28844931

Cc1cnnc(NCC(C)(C)c2ccc(F)cc2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33
ME2 P23368 1/20 0.33
ME1 P48163 1/20 0.33
ME3 Q16798 1/20 0.33
BMI1 P35226 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
TRPV1 Q8NER1 2/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM4E B2RXH2 1/20 0.31
IL1B P01584 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27898833 0.80 FPR2 (0.41) ME2ME1ME3CACNA1G
SCHEMBL28148590 0.77 GOT1 (0.39) CACNA1G
SCHEMBL17700425 0.77 HRH4 (0.38) CYP11B1CYP11B2IL1BTNF
SCHEMBL2562929 0.77 MEN1 (0.38) KMT2AMEN1IL1BTNFCACNA1G
SCHEMBL17240868 0.75 IL1B (0.36) LMNAKMT2ACYP3A4CYP2D6CYP2C9
SCHEMBL14734750 0.73 MEN1 (0.32) KMT2AHTTMEN1SMN1; SMN2IL1B
SCHEMBL21170499 0.73 KDM4E (0.40) LMNAKMT2ACYP3A4CYP2D6CYP2C9
SCHEMBL21170299 0.72 NPC1 (0.47) LMNAKMT2ACYP3A4CYP2D6CYP2C9
SCHEMBL17240865 0.71 IL1B (0.33) IL1BTNFCACNA1G
SCHEMBL2561843 0.71 MAPT (0.43) KMT2AHTTMEN1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107266419-A Specific amino pyridazine class, thing in combination, and its application method 赛特凯恩蒂克公司 2017-10-20 CN disclosed
CN-103002897-B Certain amino-pyridazines, compositions thereof, and methods of use thereof 赛特凯恩蒂克公司 2017-06-09 CN disclosed