SCHEMBL28845158

SCHEMBL28845158

N#Cc1ccc(OC=O)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.35
NSD3 Q9BZ95 1/20 0.35
CHEK1 O14757 3/20 0.34
CCR2 P41597 1/20 0.34
AR P10275 1/20 0.33
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
TRPA1 O75762 1/20 0.33
EGLN2 Q96KS0 1/20 0.33
PDE10A Q9Y233 1/20 0.32
NQO1 P15559 1/20 0.32
VHL P40337 1/20 0.32
SLC40A1 Q9NP59 1/20 0.31
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRB1 P18505 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15865529 0.74 CBFB (0.40) CHEK1NQO1ALOX5APFEN1
SCHEMBL4657354 0.74 KDM4E (0.40) POLB
SCHEMBL240556 0.74 NQO1 (0.50) PDE10ANQO1POLB
SCHEMBL1145498 0.74 NSD2 (0.38) NSD2NSD3CHEK1CCR2AR
SCHEMBL450834 0.72 ALDH1A1 (0.42) CHEK1ARKCNQ3KCNQ2EGLN2
SCHEMBL12225600 0.72 CHRNA3 (0.41)
SCHEMBL22120385 0.72 NSD2 (0.49) NSD2NSD3CHEK1MMP3
SCHEMBL13513874 0.72 KMT2A (0.42)
SCHEMBL195649 0.71 CA2 (0.48) MMP2MMP3POLB
SCHEMBL28893504 0.71 NQO1 (0.50) NSD2NSD3CHEK1NQO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106795147-A Cyclopropyl fused thiazine-2-amine compounds as beta-secretase inhibitors and methods of use 美国安进公司 2017-05-31 CN disclosed