SCHEMBL28845680

SCHEMBL28845680

O=C(NCCO)c1ccc(Nc2ccnc3cc(C(F)(F)F)ccc23)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAK O14976 3/20 0.51
DNMT1 P26358 3/20 0.48
DNMT3A Q9Y6K1 2/20 0.48
HDAC3 O15379 1/20 0.48
ACHE P22303 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
DNMT3L Q9UJW3 1/20 0.48
GPR52 Q9Y2T5 3/20 0.47
GSK3A P49840 4/20 0.47
GSK3B P49841 4/20 0.47
CLK4 Q9HAZ1 4/20 0.47
AURKB Q96GD4 3/20 0.47
PRKD3 O94806 2/20 0.47
MAP4K4 O95819 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28845632 0.94 GAK (0.49) GAKDNMT1DNMT3AHDAC3ACHE
SCHEMBL28845671 0.91 GAK (0.53) GAKDNMT1DNMT3AHDAC3ACHE
SCHEMBL28845651 0.90 GPR52 (0.54) GAKDNMT1DNMT3AGPR52GSK3A
SCHEMBL28845677 0.88 GAK (0.54) GAKDNMT1DNMT3AHDAC3ACHE
SCHEMBL28845682 0.85 DNMT1 (0.54) GAKDNMT1DNMT3AHDAC3ACHE
SCHEMBL10664310 0.84 GAK (0.57) GAKDNMT1DNMT3AHDAC3ACHE
SCHEMBL28845643 0.84 GPR52 (0.59) GAKDNMT1DNMT3AGPR52GSK3A
Hydrochloric Acid SCHEMBL11735917 0.84 GAK (0.56) GAKDNMT1DNMT3AHDAC3ACHE
SCHEMBL1867232 0.84 TRPV1 (0.49) RIPK2
Hydrochloric Acid SCHEMBL11523664 0.83 GAK (0.56) GAKDNMT1DNMT3AHDAC3ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN claimed
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN disclosed
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN disclosed