SCHEMBL28845643

SCHEMBL28845643

O=C(NCCCO)c1cccc(Nc2ccnc3cc(C(F)(F)F)ccc23)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 4/20 0.59
MRGPRX4 Q96LA9 1/20 0.49
DNMT1 P26358 1/20 0.49
DNMT3A Q9Y6K1 1/20 0.49
EPHX2 P34913 1/20 0.46
GAK O14976 2/20 0.46
GSK3A P49840 3/20 0.46
GSK3B P49841 3/20 0.46
CLK4 Q9HAZ1 2/20 0.46
PRKD3 O94806 1/20 0.46
MAP4K4 O95819 1/20 0.46
MARK3 P27448 1/20 0.46
KDR P35968 1/20 0.46
MAPKAPK2 P49137 1/20 0.46
PRKCZ Q05513 1/20 0.46
PRKAA1 Q13131 1/20 0.46
PAK1 Q13153 1/20 0.46
STK3 Q13188 1/20 0.46
TAOK1 Q7L7X3 1/20 0.46
HIPK4 Q8NE63 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28845651 0.94 GPR52 (0.54) GPR52MRGPRX4DNMT1DNMT3AGAK
SCHEMBL28845632 0.90 GAK (0.49) GPR52MRGPRX4DNMT1DNMT3AEPHX2
SCHEMBL28845687 0.90 ALDH1A1 (0.57) GPR52MRGPRX4DNMT1DNMT3AGAK
SCHEMBL28845637 0.87 DNMT1 (0.52) GPR52MRGPRX4DNMT1DNMT3AGAK
SCHEMBL28845665 0.87 CCNC (0.51) GPR52DNMT1DNMT3AGAKGSK3A
SCHEMBL28845680 0.84 GAK (0.51) GPR52DNMT1DNMT3AGAKGSK3A
SCHEMBL28845675 0.83 DNMT1 (0.68) DNMT1DNMT3AGAKGSK3AGSK3B
SCHEMBL28845630 0.83 KMT2A (0.46) GPR52GAKGSK3AGSK3BCLK4
SCHEMBL29200469 0.82 GAK (0.55) DNMT1DNMT3AGAKGSK3AGSK3B
SCHEMBL28845648 0.82 NPSR1 (0.56) GPR52MRGPRX4DNMT1DNMT3AGAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN claimed
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN disclosed
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN disclosed