SCHEMBL28845689

SCHEMBL28845689

CCOc1ccc(N2CCN(C(=O)c3cccc(Nc4ccnc5cc(C(F)(F)F)ccc45)c3)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.52
ALDH1A1 P00352 1/20 0.52
GAA P10253 1/20 0.52
ALOX15 P16050 1/20 0.52
MAPK1 P28482 1/20 0.52
HTT P42858 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
LMNA P02545 2/20 0.48
TP53 P04637 1/20 0.48
GPR52 Q9Y2T5 2/20 0.46
PDGFRB P09619 1/20 0.46
MAPKAPK2 P49137 2/20 0.46
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
GAK O14976 2/20 0.44
KMT2A Q03164 1/20 0.44
THRB P10828 1/20 0.43
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
SCN9A Q15858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28845629 0.91 MAPKAPK2 (0.49) MAPTALDH1A1GAAALOX15HTT
SCHEMBL30771663 0.91 MAPKAPK2 (0.49) MAPTALDH1A1MAPK1HTTLMNA
SCHEMBL29200486 0.91 MAPKAPK2 (0.49) MAPTALDH1A1MAPK1HTTLMNA
SCHEMBL28845661 0.91 SCN9A (0.48) MAPTGAAHTTLMNAGPR52
SCHEMBL28845640 0.90 MAPKAPK2 (0.49) GPR52MAPKAPK2GAKKMT2ADRD2
SCHEMBL28845636 0.89 DRD2 (0.51) MAPTGAAMAPK1HTTTDP1
SCHEMBL28845652 0.88 RAD52 (0.49) MAPTALDH1A1MAPK1HTTLMNA
SCHEMBL29809902 0.86 ABL1 (0.50) MAPTGPR52MAPKAPK2KMT2ASCN9A
SCHEMBL28845642 0.86 ABL1 (0.50) MAPTGPR52MAPKAPK2KMT2ASCN9A
SCHEMBL29809938 0.83 HPGD (0.56) ALDH1A1LMNAGPR52MAPKAPK2GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN disclosed
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN disclosed