SCHEMBL29200486

SCHEMBL29200486

O=C(c1cccc(Nc2ccnc3cc(C(F)(F)F)ccc23)c1)N1CCN(c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 2/20 0.49
GPR52 Q9Y2T5 2/20 0.49
SCN9A Q15858 1/20 0.48
POLB P06746 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
EPHX2 P34913 3/20 0.47
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
ABL1 P00519 2/20 0.46
BCR P11274 2/20 0.46
PDGFRB P09619 1/20 0.46
NAMPT P43490 1/20 0.45
KDM4E B2RXH2 3/20 0.45
MAPT P10636 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30771663 1.00 MAPKAPK2 (0.49) MAPKAPK2GPR52SCN9APOLBSMN1; SMN2
SCHEMBL28845636 0.96 DRD2 (0.51) MAPKAPK2GPR52POLBSMN1; SMN2MEN1
SCHEMBL28845640 0.95 MAPKAPK2 (0.49) MAPKAPK2GPR52SCN9APOLBSMN1; SMN2
SCHEMBL28845652 0.95 RAD52 (0.49) MAPKAPK2GPR52POLBSMN1; SMN2MEN1
SCHEMBL28845661 0.93 SCN9A (0.48) MAPKAPK2GPR52SCN9APOLBSMN1; SMN2
SCHEMBL28845642 0.91 ABL1 (0.50) MAPKAPK2GPR52SCN9APOLBSMN1; SMN2
SCHEMBL29809902 0.91 ABL1 (0.50) MAPKAPK2GPR52SCN9APOLBSMN1; SMN2
SCHEMBL28845689 0.91 MAPT (0.52) MAPKAPK2GPR52SCN9AKMT2ADRD2
SCHEMBL29809938 0.89 HPGD (0.56) MAPKAPK2GPR52POLBMEN1KMT2A
SCHEMBL29809947 0.87 ADRB2 (0.49) MAPKAPK2GPR52POLBEPHX2ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN disclosed