SCHEMBL28845697

SCHEMBL28845697

Cc1cccc(N2CCN(c3cccc(C(=O)Nc4ccnc5cc(C(F)(F)F)ccc45)c3)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.51
KDM4E B2RXH2 1/20 0.51
TP53 P04637 2/20 0.50
GAA P10253 1/20 0.50
GSK3A P49840 4/20 0.48
GSK3B P49841 4/20 0.48
CLK4 Q9HAZ1 3/20 0.48
KDR P35968 3/20 0.48
PRKD3 O94806 2/20 0.48
MAP4K4 O95819 2/20 0.48
AURKB Q96GD4 2/20 0.48
PRKD2 Q9BZL6 2/20 0.48
MARK3 P27448 1/20 0.48
MAPKAPK2 P49137 1/20 0.48
PRKCZ Q05513 1/20 0.48
PRKAA1 Q13131 1/20 0.48
PAK1 Q13153 1/20 0.48
STK3 Q13188 1/20 0.48
TAOK1 Q7L7X3 1/20 0.48
HIPK4 Q8NE63 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29809960 1.00 MAPT (0.51) MAPTKDM4ETP53GAAGSK3A
SCHEMBL28845694 0.86 TP53 (0.52) MAPTKDM4ETP53GAAGSK3A
SCHEMBL29809952 0.86 TP53 (0.52) MAPTKDM4ETP53GAAGSK3A
SCHEMBL28845642 0.84 ABL1 (0.50) MAPTMAPKAPK2RAB9AKMT2APHGDH
SCHEMBL29809902 0.84 ABL1 (0.50) MAPTMAPKAPK2RAB9AKMT2APHGDH
SCHEMBL29809955 0.80 MEN1 (0.61) MAPTGSK3AGSK3BCLK4KDR
SCHEMBL28845693 0.80 MEN1 (0.61) MAPTGSK3AGSK3BCLK4KDR
SCHEMBL28845640 0.77 MAPKAPK2 (0.49) MAPKAPK2KMT2APHGDHABL1MEN1
SCHEMBL28845668 0.76 GAA (0.60) MAPTGAAGSK3AGSK3BCLK4
SCHEMBL28845644 0.76 KMT2A (0.52) MAPTMAPKAPK2KMT2APHGDHMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN disclosed
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN disclosed