SCHEMBL28845830

SCHEMBL28845830

CN1CCN(c2ccc(-c3ccoc3)cc2-c2ncc(N)c(N)n2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
WDR5 P61964 1/20 0.49
HRH4 Q9H3N8 2/20 0.49
HRH1 P35367 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49
HDAC3 O15379 2/20 0.48
HDAC2 Q92769 2/20 0.48
CYP1A2 P05177 5/20 0.46
CYP2D6 P10635 4/20 0.46
ALDH1A1 P00352 3/20 0.46
CYP3A4 P08684 3/20 0.46
MEN1 O00255 2/20 0.46
USP2 O75604 2/20 0.46
CLK4 Q9HAZ1 2/20 0.46
HIF1A Q16665 1/20 0.46
ALOX15 P16050 3/20 0.46
HSD17B10 Q99714 2/20 0.46
CYP2C19 P33261 1/20 0.44
HTR1A P08908 2/20 0.42
DRD2 P14416 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28845808 0.84 WDR5 (0.49) KMT2AWDR5HRH4CYP1A2CYP2D6
SCHEMBL28291860 0.84 WDR5 (0.47) KMT2AWDR5HRH4HDAC2CYP1A2
SCHEMBL28953596 0.78 CYP1A2 (0.49) KMT2AHRH4HRH3CYP1A2CYP2D6
SCHEMBL28845844 0.74 WDR5 (0.48) KMT2AWDR5HRH4CYP1A2CYP2D6
SCHEMBL4620360 0.73 FYN (0.69) KMT2AHRH4HRH1HRH3HDAC3
SCHEMBL24166935 0.66 WDR5 (1.00) KMT2AWDR5
SCHEMBL29545139 0.66 WDR5 (1.00) KMT2AWDR5
SCHEMBL1030754 0.66 HRH4 (1.00) KMT2AHRH4HRH1HRH3CYP1A2
SCHEMBL28953598 0.66 HRH4 (0.42) HRH4ALDH1A1DRD2
SCHEMBL20181651 0.65 HDAC2 (1.00) HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734674-B Aniline WDR5 protein-protein interaction inhibitor and preparation method and application thereof 中国药科大学 2022-08-26 CN disclosed