SCHEMBL28845844

SCHEMBL28845844

CN1CCN(c2ccc([N+](=O)[O-])cc2-c2ncc(N)c(N)n2)CC1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 7/20 0.48
KMT2A Q03164 6/20 0.48
ALDH1A1 P00352 7/20 0.47
LMNA P02545 3/20 0.47
GAA P10253 2/20 0.47
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
MEN1 O00255 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HRH4 Q9H3N8 1/20 0.45
KDM4E B2RXH2 1/20 0.44
HTT P42858 2/20 0.43
SIRT6 Q8N6T7 1/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28845821 0.87 MEN1 (0.49) KMT2AALDH1A1LMNAGAAMEN1
SCHEMBL29890962 0.87 WDR5 (0.48) WDR5KMT2AALDH1A1LMNACYP1A2
SCHEMBL28845825 0.87 WDR5 (0.48) WDR5KMT2AALDH1A1LMNACYP1A2
SCHEMBL29890986 0.82 ALDH1A1 (0.54) WDR5KMT2AALDH1A1LMNAGAA
SCHEMBL28845797 0.81 KMT2A (0.52) WDR5KMT2AALDH1A1LMNAGAA
SCHEMBL28845817 0.78 WDR5 (0.52) WDR5KMT2AALDH1A1LMNAGAA
SCHEMBL1969337 0.77 SIRT6 (0.58) WDR5KMT2AALDH1A1LMNAGAA
SCHEMBL28291860 0.77 WDR5 (0.47) WDR5KMT2ACYP1A2CYP2C19HRH4
SCHEMBL28845808 0.77 WDR5 (0.49) WDR5KMT2AALDH1A1CYP1A2CYP3A4
SCHEMBL28845803 0.75 TDP1 (0.44) KMT2AALDH1A1LMNAGAACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734674-B Aniline WDR5 protein-protein interaction inhibitor and preparation method and application thereof 中国药科大学 2022-08-26 CN disclosed