SCHEMBL28847446

SCHEMBL28847446

CC(c1cc(N)c(N)c(Br)c1)C(C(N)=O)N1CCOCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.44
CYP3A4 P08684 2/20 0.35
HIF1A Q16665 1/20 0.35
ALDH1A1 P00352 8/20 0.33
TSHR P16473 3/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KMT2A Q03164 3/20 0.32
HPGD P15428 2/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
F2 P00734 1/20 0.31
F7 P08709 1/20 0.31
HTT P42858 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
MAPK1 P28482 1/20 0.31
GLA P06280 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28847499 0.85 ALDH1A1 (0.37) AAK1CYP3A4ALDH1A1SMN1; SMN2KMT2A
SCHEMBL28847473 0.81 AAK1 (0.41) AAK1CYP3A4HIF1AALDH1A1TSHR
SCHEMBL28847447 0.74 MAPT (0.43) ALDH1A1SMN1; SMN2KMT2ALMNAMAPT
SCHEMBL28847427 0.73 AAK1 (0.39) AAK1CYP3A4HIF1AALDH1A1TSHR
SCHEMBL28847388 0.73 MAPT (0.41) AAK1ALDH1A1SMN1; SMN2KMT2ALMNA
SCHEMBL28847456 0.72 NPC1 (0.46) ALDH1A1TSHRSMN1; SMN2KMT2ALMNA
SCHEMBL28847442 0.71 KDM1A (0.41) AAK1HIF1AALDH1A1SMN1; SMN2KMT2A
SCHEMBL23525085 0.70 AAK1 (0.48) AAK1ALDH1A1KMT2A
SCHEMBL23525084 0.70 AAK1 (0.48) AAK1ALDH1A1KMT2A
SCHEMBL28847449 0.69 MAPT (0.41) CYP3A4ALDH1A1CYP2C19LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115087655-A Benzimidazole derivatives 辉瑞公司 2022-09-20 CN disclosed