SCHEMBL28849571

SCHEMBL28849571

O=CNc1ccc2c(c1)C=CC2

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.32
OPRD1 P41143 2/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28062192 0.98 ALDH1A1 (0.35) ALDH1A1LMNAOPRD1CA1CA2
SCHEMBL24493269 0.76 EGFR (0.30) CA1CA2
SCHEMBL30950742 0.74 RAB9A (0.37) ALDH1A1
SCHEMBL28122675 0.73
SCHEMBL29561757 0.72 ALDH1A1 (0.38) ALDH1A1
SCHEMBL19633072 0.71
SCHEMBL28178883 0.71 ALDH1A1 (0.33) ALDH1A1OPRD1
SCHEMBL28219230 0.71 ALDH1A1 (0.33) ALDH1A1
SCHEMBL27761248 0.70 ALDH1A1 (0.36) ALDH1A1
SCHEMBL275807 0.70 CA1 (0.33) CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107205972-A Substituted N- (2- (amino) -2-oxoethyl) benzamide inhibitors of autotaxin and their preparation and use in the treatment of LPA-dependent or LPA-mediated diseases X-RX股份有限公司 2017-09-26 CN claimed
CN-107205972-A Substituted N- (2- (amino) -2-oxoethyl) benzamide inhibitors of autotaxin and their preparation and use in the treatment of LPA-dependent or LPA-mediated diseases X-RX股份有限公司 2017-09-26 CN disclosed