SCHEMBL28850451

SCHEMBL28850451

CCC1CCc2c(ccc3c2CCc2ccccc2-3)C1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 15/20 0.39
HTR1A P08908 14/20 0.39
CES1 P23141 1/20 0.36
CYP19A1 P11511 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28086055 0.83 CYP19A1 (0.46) HTR1ACYP19A1
SCHEMBL28838816 0.81 HTR7 (0.43) HTR7HTR1ACES1
SCHEMBL20131349 0.77 HTR7 (0.63) HTR7HTR1A
SCHEMBL20131348 0.77 HTR7 (0.63) HTR7HTR1A
SCHEMBL28210257 0.75 DAPK3 (0.41) HTR7HTR1ACES1CYP19A1
SCHEMBL15412764 0.73 CYP19A1 (0.37) CYP19A1
SCHEMBL599314 0.72 CYP19A1 (0.54) HTR1ACYP19A1
SCHEMBL28167514 0.72 CYP19A1 (0.46) HTR1ACYP19A1
SCHEMBL27697275 0.72 DYRK1A (0.35) HTR7HTR1ACES1
SCHEMBL13448455 0.71 CYP19A1 (0.41) HTR7HTR1ACYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107074861-A 9H pyrimido [4,5-B ] indoles and related analogs as BET bromodomain inhibitors 密执安大学评议会 2017-08-18 CN disclosed