SCHEMBL28852844

SCHEMBL28852844

CS(=O)(=O)N(C#Cc1ccccc1)CC(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 7/20 0.40
NPC1 O15118 1/20 0.40
MTOR P42345 1/20 0.40
RAB9A P51151 1/20 0.40
PTPN1 P18031 1/20 0.39
NR1H2 P55055 7/20 0.38
RORC P51449 3/20 0.36
RORA P35398 1/20 0.36
RORB Q92753 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
APP P05067 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28852909 0.78 ALDH1A1 (0.42) NPC1MTORRAB9ACA2
SCHEMBL28389232 0.71 NPC1 (0.48) NPC1MTORRAB9APTPN1NR1H2
SCHEMBL28852821 0.68 NPC1 (0.42) NPC1MTORRAB9APTPN1CA12
SCHEMBL28852773 0.66 NPC1 (0.40) NPC1MTORRAB9APTPN1NR1H2
SCHEMBL10699281 0.64 APP (0.48) NPC1MTORRAB9ANPSR1APP
SCHEMBL28218124 0.64 NR1I2 (0.56) NR1I2NR1H2RORCRORARORB
SCHEMBL28852744 0.64 VCP (0.41) NPC1MTORRAB9ANR1H2CA12
SCHEMBL28852810 0.64 NPC1 (0.41) NPC1MTORRAB9APTPN1CA12
Diphenylacetylene SCHEMBL27721387 0.63 APP (0.60) NPC1MTORRAB9ACA12CA1
SCHEMBL23036810 0.63 CNR2 (0.55) NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113200891-B Preparation method of cis-N-styryl amide derivative 华侨大学 2022-09-30 CN claimed
CN-113200891-A Preparation method of cis-N-styryl amide derivative 华侨大学 2021-08-03 CN claimed
CN-113200891-B Preparation method of cis-N-styryl amide derivative 华侨大学 2022-09-30 CN disclosed
CN-113200891-A Preparation method of cis-N-styryl amide derivative 华侨大学 2021-08-03 CN disclosed