SCHEMBL28857604

SCHEMBL28857604

Cc1cc(C)n(Cc2ccc(C(=O)Nc3ccc(Br)cc3C)cc2)n1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.72
POLB P06746 1/20 0.72
GAA P10253 1/20 0.57
RAB9A P51151 1/20 0.57
CYP3A4 P08684 1/20 0.56
MAPT P10636 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
STAT3 P40763 1/20 0.56
HTT P42858 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
PTGDR2 Q9Y5Y4 4/20 0.50
TSHR P16473 1/20 0.50
DHODH Q02127 1/20 0.50
ALDH1A1 P00352 1/20 0.49
HDAC3 O15379 4/20 0.49
HDAC4 P56524 4/20 0.49
HDAC1 Q13547 4/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28857585 0.88 LMNA (0.66) LMNAPOLBGAARAB9ACYP3A4
SCHEMBL28857626 0.88 PTGDR2 (0.58) LMNAPOLBGAARAB9ACYP3A4
SCHEMBL28857612 0.87 GAA (0.57) LMNAPOLBGAARAB9ACYP3A4
SCHEMBL28857646 0.84 LMNA (1.00) LMNAPOLBGAAHTTSMN1; SMN2
SCHEMBL28955070 0.81 LMNA (0.64) LMNAPOLBRAB9ACYP3A4MAPT
SCHEMBL28857580 0.80 LMNA (0.66) LMNAPOLBGAARAB9AMAPT
SCHEMBL213450 0.79 HDAC1 (0.60) LMNAGAARAB9ACYP3A4MAPT
SCHEMBL28857591 0.78 HIF1A (0.60) LMNAPOLBGAARAB9AMAPT
SCHEMBL31462454 0.76 LMNA (0.62) LMNAPOLBGAARAB9ACYP3A4
SCHEMBL28857636 0.76 LMNA (0.81) LMNAPOLBGAAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115160269-A Arylcarboxamide derivatives as positive allosteric modulators of NMDAR 北京大学 2022-10-11 CN claimed
CN-115160269-A Arylcarboxamide derivatives as positive allosteric modulators of NMDAR 北京大学 2022-10-11 CN disclosed