Trimethobenzamide

Trimethobenzamide

SCHEMBL28858

COc1cc(C(=O)NCc2ccc(OCCN(C)C)cc2)cc(OC)c1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 1.00
DRD3 P35462 2/20 1.00
LMNA P02545 2/20 1.00
ACHE P22303 1/20 1.00
SLC6A2 P23975 1/20 1.00
CYP2C19 P33261 1/20 1.00
KCNH2 Q12809 1/20 1.00
SMN1; SMN2 Q16637 5/20 0.98
MAPK1 P28482 1/20 0.98
HRH3 Q9Y5N1 1/20 0.80
BRD4 O60885 1/20 0.58
KMT2A Q03164 1/20 0.58
ALDH1A1 P00352 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.55
HPGD P15428 2/20 0.54
NPC1 O15118 1/20 0.52
PKM P14618 1/20 0.52
KDM4E B2RXH2 1/20 0.50
RAB9A P51151 1/20 0.50
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trimethobenzamide SCHEMBL6683399 1.00 DRD2 (1.00) DRD2DRD3LMNAACHESLC6A2
Trimethobenzamide SCHEMBL4586290 0.99 DRD2 (0.98) DRD2DRD3LMNAACHESLC6A2
Trimethobenzamide SCHEMBL4586216 0.99 SMN1; SMN2 (1.00) DRD2DRD3LMNAACHESLC6A2
Trimethobenzamide SCHEMBL4586062 0.99 DRD2 (0.98) DRD2DRD3LMNAACHESLC6A2
Trimethobenzamide SCHEMBL41339 0.99 SMN1; SMN2 (1.00) DRD2DRD3LMNAACHESLC6A2
Trimethobenzamide SCHEMBL3059009 0.98 DRD2 (0.96) DRD2DRD3LMNAACHESLC6A2
Trimethobenzamide SCHEMBL4586023 0.97 DRD2 (0.94) DRD2DRD3LMNAACHESLC6A2
Trimethobenzamide SCHEMBL4586233 0.96 DRD2 (0.92) DRD2DRD3LMNAACHESLC6A2
Itopride SCHEMBL311309 0.89 DRD2 (1.00) DRD2DRD3LMNAACHESLC6A2
Itopride SCHEMBL554675 0.88 DRD2 (0.98) DRD2DRD3LMNAACHESLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6736 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4731194-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING AN ACTIVE AGENT CSP Technologies, Inc. (US) 2026-04-29 EP claimed
US-20260076872-A1 POLYMER VIALS WITH SUBSTANTIALLY FLAT BOTTOMS AND INJECTION STRETCH BLOW MOLDING METHODS FOR MAKING THE SAME SIO2 MEDICAL PRODUCTS LLC (US) 2026-03-19 US claimed
WO-2025264260-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING AN ACTIVE AGENT CSP TECHNOLOGIES, INC. (US) 2025-12-26 WO claimed
US-20250259704-A1 SYSTEMS AND METHODS FOR CELL-FREE ITERATIVE SITE SATURATION MUTAGENESIS AND ITS APPLICATION FOR THE DIRECTED EVOLUTION OF ENZYMES CATALYZING UNNATURAL REACTIONS U.S. DEPARTMENT OF ENERGY 2025-08-14 US claimed
US-20250242092-A1 SiOx BARRIER FOR PHARMACEUTICAL PACKAGE AND COATING PROCESS SIO2 MEDICAL PRODUCTS INC (US) 2025-07-31 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-12310934-B2 Methods of treatment of spontaneous preterm birth THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-05-27 US claimed
US-12257371-B2 SiOx barrier for pharmaceutical package and coating process SIO2 MEDICAL PRODUCTS, LLC (US) 2025-03-25 US claimed
WO-2024263560-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING AN ACTIVE AGENT CSP TECHNOLOGIES, INC. (US) 2024-12-26 WO claimed
US-20240366639-A1 HETEROCYCLIC GLP-1 AGONISTS GASHERBRUM BIO INC (US) 2024-11-07 US claimed
US-5288498-A Compositions of oral nondissolvable matrixes for transmucosal administration of medicaments UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 1994-02-22 US claimed
EP-0487520-A4 COMPRESSED POWDER MEDICAMENTS 1992-08-12 EP claimed
US-5132114-A Compositions and methods of manufacture of compressed powder medicaments UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 1992-07-21 US claimed
EP-0487520-A1 COMPRESSED POWDER MEDICAMENTS. ANESTA CORP (US) 1992-06-03 EP claimed
EP-0201537-B1 NOVEL USE OF ANTI-NAUSEA AND ANTI-EMETIC PHARMAZEUTICAL AGENTS. NASTECH PHARMACEUTICAL COMPANY, INC. (US) 1992-04-29 EP claimed
WO-1991003099-A1 COMPRESSED POWDER MEDICAMENTS ANESTA CORPORATION (US) 1991-03-07 WO claimed
US-4729997-A ANTIEMETICS, ANTIHISTAMINES NASTECH PHARMACEUTICAL CO., INC. (US) 1988-03-08 US claimed
EP-0201537-A4 NOVEL USE OF ANTI-NAUSEA AND ANTI-EMETIC PHARMAZEUTICAL AGENTS. NASTECH PHARM CO (US) 1987-07-06 EP claimed
EP-0201537-A1 NOVEL USE OF ANTI-NAUSEA AND ANTI-EMETIC PHARMAZEUTICAL AGENTS. NASTECH PHARM CO (US) 1986-11-20 EP claimed
WO-1986002553-A1 NOVEL METHOD OF ADMINISTERING ANTI-NAUSEA AND ANTI-EMETIC PHARMACEUTICAL AGENTS AND NOVEL DOSAGE FORMS CONTAINING SAME NASTECH PHARMACEUTICAL COMPANY, INC. (US) 1986-05-09 WO claimed