SCHEMBL28858007

SCHEMBL28858007

NC(=O)c1cc2cc(-c3ccc(C(F)(F)F)cc3)ccc2[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 4/20 0.49
HPN P05981 1/20 0.49
DHODH Q02127 1/20 0.48
HRH4 Q9H3N8 1/20 0.47
SLC6A2 P23975 1/20 0.46
PLD2 O14939 1/20 0.45
PLD1 Q13393 1/20 0.45
MMP2 P08253 1/20 0.45
MMP13 P45452 1/20 0.45
MMP14 P50281 1/20 0.45
PARP1 P09874 1/20 0.45
KIF11 P52732 3/20 0.45
ABCB1 P08183 1/20 0.43
MAP2K4 P45985 1/20 0.43
CHEK2 O96017 1/20 0.43
KDM4E B2RXH2 2/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
PDPK1 O15530 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30314640 0.88 HRH4 (0.58) P2RY14HRH4PLD2PLD1MMP2
SCHEMBL28208771 0.84 KDM4E (0.55) HPNHRH4MMP2MMP13MMP14
SCHEMBL28207999 0.82 KDM4E (0.60) MMP2MMP13MMP14ABCB1CHEK2
SCHEMBL26306635 0.79 HRH4 (0.46) P2RY14HRH4SLC6A2PLD2PLD1
SCHEMBL333745 0.79 MMP13 (0.74) MMP2MMP13MMP14KDM4EGAA
SCHEMBL29619366 0.79 P2RY14 (0.50) P2RY14HRH4PLD2PLD1PARP1
SCHEMBL11552360 0.78 HRH4 (0.45) P2RY14HRH4PLD2PLD1MMP2
SCHEMBL22525900 0.76 PTPN1 (0.54) P2RY14HRH4PLD2PLD1KDM4E
SCHEMBL13554437 0.76 MMP2 (0.46) HRH4MMP2MMP13KIF11KDM4E
SCHEMBL16599412 0.75 HRH4 (0.60) HRH4PLD2PLD1KDM4EPDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555763-B indole-carboxamide derivatives 豪夫迈·罗氏有限公司 2018-04-17 CN claimed
CN-105555763-B indole-carboxamide derivatives 豪夫迈·罗氏有限公司 2018-04-17 CN disclosed