SCHEMBL28861602

SCHEMBL28861602

COc1ccc(-c2nc3c(N)nc(N)nc3[nH]2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.51
DHFR P00374 5/20 0.47
HEXA P06865 1/20 0.47
HEXB P07686 1/20 0.47
PARP1 P09874 3/20 0.46
PLA2G2A P14555 1/20 0.46
ALOX15 P16050 1/20 0.46
PTGS2 P35354 1/20 0.46
ALDH1A1 P00352 3/20 0.46
NPC1 O15118 2/20 0.46
PKM P14618 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
RAB9A P51151 1/20 0.46
TNKS O95271 2/20 0.45
TNKS2 Q9H2K2 2/20 0.45
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45
POLB P06746 1/20 0.45
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL4273194 0.86 KDM4E (0.49) KDM4EDHFRPARP1PLA2G2AALOX15
SCHEMBL3121094 0.85 KDM4E (0.48) KDM4EDHFRPARP1PLA2G2AALOX15
SCHEMBL27870414 0.83 PIK3CG (0.57) DHFRPARP1NPC1PKMRAB9A
SCHEMBL27870416 0.83 HEXA (0.43) DHFRHEXAHEXBPARP1TNKS
SCHEMBL15756441 0.82 MAP4K4 (0.48) KDM4EPARP1PLA2G2AALOX15PTGS2
SCHEMBL27886649 0.80 MMP2 (0.41) KDM4EDHFRPARP1NPC1RAB9A
SCHEMBL27870415 0.80 MGAM (0.44) KDM4EDHFRPARP1ALDH1A1NPC1
SCHEMBL2947301 0.80 PDE2A (0.48) KDM4EALDH1A1
SCHEMBL27886638 0.80 ALDH1A1 (0.47) KDM4EDHFRPARP1ALDH1A1NPC1
SCHEMBL28230094 0.78 PARP1 (0.45) KDM4EPARP1ALDH1A1NPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108371662-B Application of five-membered heterocyclic pyrimidine compound 中国药科大学 2023-03-03 CN claimed
CN-108371662-A A kind of application of five-ring heterocycles miazines compound 中国药科大学 2018-08-07 CN claimed
CN-108371662-A A kind of application of five-ring heterocycles miazines compound 中国药科大学 2018-08-07 CN disclosed