SCHEMBL2947301

SCHEMBL2947301

COc1ccc(-c2nc3c(N)nc(N)nc3[nH]2)c(OC)c1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.48
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
GFER P55789 1/20 0.45
SLC2A1 P11166 1/20 0.45
KDM4E B2RXH2 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
EGFR P00533 1/20 0.43
TYMS P04818 1/20 0.43
KDR P35968 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28861590 0.83 SLC2A1 (0.62) ALDH1A1GAASLC2A1
SCHEMBL2954598 0.82 DHFR (0.43) SLC2A1CYP3A4
SCHEMBL28861602 0.80 KDM4E (0.51) ALDH1A1KDM4E
SCHEMBL7968435 0.79 PDE2A (0.50) PDE2AALDH1A1GAAMAPK1HTT
SCHEMBL27870414 0.78 PIK3CG (0.57) HTTCYP1A2
SCHEMBL2952943 0.78 MAP2K7 (0.45) CYP3A4
SCHEMBL1966500 0.77 HSP90AA1 (0.56) EGFRKDR
SCHEMBL10846727 0.76 PDE2A (0.62) PDE2AALDH1A1GAAMAPK1HTT
SCHEMBL10685704 0.76 PDE2A (0.50) PDE2AALDH1A1GAAMAPK1HTT
SCHEMBL2946218 0.75 CHEK1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed