SCHEMBL28862

SCHEMBL28862

Cn1cccc1C(=O)N1CCN(C(=O)Nc2ccc(N3CCC(C4CCCCN4)CC3=C=O)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 15/20 0.54
CYP3A4 P08684 4/20 0.44
USP2 O75604 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 3/20 0.41
MAPK1 P28482 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27590 0.82 HPGDS (0.59) HPGDSCYP3A4USP2SMN1; SMN2ALDH1A1
SCHEMBL28861 0.74 HPGDS (0.71) HPGDSCYP3A4USP2SMN1; SMN2ALDH1A1
SCHEMBL27841 0.71 HPGDS (1.00) HPGDSCYP3A4USP2SMN1; SMN2ALDH1A1
SCHEMBL27589 0.68 HPGDS (1.00) HPGDS
Morpholine SCHEMBL28316 0.67 HPGDS (0.59) HPGDSCYP3A4USP2SMN1; SMN2ALDH1A1
SCHEMBL27787 0.67 HPGDS (1.00) HPGDS
SCHEMBL29363 0.66 HPGDS (1.00) HPGDS
SCHEMBL28315 0.65 HPGDS (1.00) HPGDSCYP3A4
SCHEMBL28755 0.65 HPGDS (1.00) HPGDS
SCHEMBL23017395 0.64 HPGDS (0.73) HPGDSCYP3A4USP2SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2407466-A1 PIPERAZINE COMPOUND CAPABLE OF INHIBITING PROSTAGLANDIN D SYNTHASE Taiho Pharmaceutical Co., Ltd. (JP) 2012-01-18 EP disclosed