SCHEMBL28863147

SCHEMBL28863147

CN(C)CCCN1CCc2ccccc21

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.82
ALDH1A1 P00352 5/20 0.82
LMNA P02545 4/20 0.82
KDM4E B2RXH2 4/20 0.82
PTK2B Q14289 1/20 0.82
ESR2 Q92731 1/20 0.82
SLC6A4 P31645 8/20 0.67
HRH1 P35367 5/20 0.67
SLC22A1 O15245 3/20 0.67
CHRM2 P08172 3/20 0.67
CHRM4 P08173 3/20 0.67
HTR1A P08908 3/20 0.67
CHRM5 P08912 3/20 0.67
CYP2D6 P10635 3/20 0.67
CHRM1 P11229 3/20 0.67
DRD2 P14416 3/20 0.67
ADRA2B P18089 3/20 0.67
ADRA2C P18825 3/20 0.67
CHRM3 P20309 3/20 0.67
DRD1 P21728 3/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7680979 0.90 ALDH1A1 (1.00) MAPTALDH1A1LMNAKDM4EPTK2B
SCHEMBL30298406 0.88 MAPT (0.64) MAPTALDH1A1LMNAKDM4EPTK2B
SCHEMBL10993180 0.85 ALDH1A1 (0.64) MAPTALDH1A1LMNAKDM4EPTK2B
SCHEMBL10983074 0.85 ALDH1A1 (0.64) MAPTALDH1A1LMNAKDM4EPTK2B
SCHEMBL3642723 0.81 ALDH1A1 (0.72) MAPTALDH1A1LMNAKDM4EPTK2B
SCHEMBL1450332 0.81 ALDH1A1 (0.82) MAPTALDH1A1LMNAKDM4EPTK2B
SCHEMBL7940135 0.80 ALDH1A1 (1.00) MAPTALDH1A1LMNAKDM4EPTK2B
Imipramine SCHEMBL17004048 0.80 SLC6A4 (1.00) MAPTALDH1A1LMNAKDM4ESLC6A4
Imipramine SCHEMBL34282 0.80 SLC6A4 (1.00) MAPTALDH1A1LMNAKDM4ESLC6A4
SCHEMBL29531557 0.80 ALDH1A1 (0.70) MAPTALDH1A1LMNAKDM4EPTK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108495855-A Condesned thiazole and pyrimidine derivatives as MNK inhibitor 生命弧度公司 2018-09-04 CN disclosed