SCHEMBL28866348

SCHEMBL28866348

ON=CC1CCc2[nH]c3ccccc3c2C1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR2E1 Q9Y466 2/20 0.58
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
TP53 P04637 1/20 0.45
KDM4E B2RXH2 2/20 0.44
HTR5A P47898 1/20 0.44
NISCH Q9Y2I1 1/20 0.44
TAAR1 Q96RJ0 1/20 0.43
RB1 P06400 2/20 0.43
SSTR3 P32745 1/20 0.42
KCNH2 Q12809 1/20 0.42
SLC2A1 P11166 1/20 0.41
BRD3 Q15059 1/20 0.41
CHRNA7 P36544 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27700723 0.89 RB1 (0.52) NR2E1HTR2AHTR2CKDM4EHTR5A
SCHEMBL7066276 0.81 NR2E1 (0.63) NR2E1HTR2AHTR2CHPGDHSD17B10
SCHEMBL2515919 0.77 NR2E1 (0.67) NR2E1HTR2AHTR2CHPGDHSD17B10
SCHEMBL4288282 0.77 NR2E1 (0.67) NR2E1HTR2AHTR2CHPGDHSD17B10
SCHEMBL833503 0.74 NR2E1 (1.00) NR2E1HTR2AHTR2CHPGDHSD17B10
SCHEMBL21900686 0.74 NR2E1 (0.67) NR2E1HTR2AHTR2CHPGDHSD17B10
SCHEMBL29670383 0.74 NR2E1 (1.00) NR2E1HTR2AHTR2CHPGDHSD17B10
SCHEMBL21754250 0.74 NR2E1 (0.67) NR2E1HTR2AHTR2CHPGDHSD17B10
SCHEMBL700531 0.74 NR2E1 (1.00) NR2E1HTR2AHTR2CHPGDHSD17B10
SCHEMBL834930 0.74 NR2E1 (1.00) NR2E1HTR2AHTR2CHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110382479-A The fluoro- 3- hydroxyl propyl- 2- base ester derivative of carbamic acid 1,1,1- tri- as MAGL inhibitor 辉瑞大药厂 2019-10-25 CN disclosed
CN-110234638-A Heteroaryl phenoxy benzamide KAPPA opiates ligand 辉瑞大药厂 2019-09-13 CN disclosed
CN-110198944-A Heterocyclic ring spiroring compounds as monoacylglycerol lipase inhibitor 辉瑞大药厂 2019-09-03 CN disclosed
CN-108884093-A 6,7,8,9- tetrahydro -5H- pyrido [2,3-d] azepine * dopamine D 3 ligands 辉瑞公司 2018-11-23 CN disclosed