SCHEMBL833503

SCHEMBL833503

NC1CCc2[nH]c3ccccc3c2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR2E1 Q9Y466 1/20 1.00
HTR6 P50406 1/20 0.60
HTR1B P28222 4/20 0.59
HTR1D P28221 3/20 0.59
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
TP53 P04637 1/20 0.50
HPGD P15428 1/20 0.50
HSD17B10 Q99714 1/20 0.50
SSTR3 P32745 1/20 0.49
KCNH2 Q12809 1/20 0.49
TAAR1 Q96RJ0 1/20 0.49
RB1 P06400 2/20 0.48
EGFR P00533 1/20 0.47
IGF1R P08069 1/20 0.47
FLT4 P35916 1/20 0.47
KDR P35968 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL700531 1.00 NR2E1 (1.00) NR2E1HTR6HTR1BHTR1DHTR2A
SCHEMBL29670383 1.00 NR2E1 (1.00) NR2E1HTR6HTR1BHTR1DHTR2A
SCHEMBL834930 1.00 NR2E1 (1.00) NR2E1HTR6HTR1BHTR1DHTR2A
Hydrochloric Acid SCHEMBL7412638 0.98 NR2E1 (0.97) NR2E1HTR6HTR1BHTR1DHTR2A
SCHEMBL29991655 0.88 NR2E1 (0.79) NR2E1HTR6HTR1BHTR1DHTR2A
SCHEMBL29992005 0.88 NR2E1 (0.79) NR2E1HTR6HTR1BHTR1DHTR2A
SCHEMBL6533665 0.88 NR2E1 (0.79) NR2E1HTR6HTR1BHTR1DHTR2A
SCHEMBL4905673 0.88 NR2E1 (0.79) NR2E1HTR6HTR1BHTR1DHTR2A
Hydrochloric Acid SCHEMBL11283863 0.87 NR2E1 (0.77) NR2E1HTR6HTR1BHTR1DHTR2A
SCHEMBL8702813 0.87 NR2E1 (0.75) NR2E1HTR6HTR1BHTR1DHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117586428-A Biomass-based macromolecular ultraviolet absorber and preparation method and application thereof 浙江沛格科技有限公司 2024-02-23 CN claimed
CN-104402798-B A kind of 3-amino-1, the method for splitting of 2,3,4-tetrahydro carbazoles 杭州瑞德化工有限公司 2016-09-14 CN claimed
CN-104402798-A Resolution method for 3-amino-1, 2, 3, 4-tetrahydrocarbazole HANGZHOU READ CHEMICAL CO LTD 2015-03-11 CN claimed
EP-4710923-A2 INDOLE AHR INHIBITORS AND USES THEREOF Ikena Oncology, Inc. (US) 2026-03-18 EP disclosed
EP-3612030-B1 INDOLE AHR INHIBITORS AND USES THEREOF IKENA ONCOLOGY INC (US) 2025-12-24 EP disclosed
US-20250129092-A1 COMPOUNDS USEFUL IN MODULATION OF AHR SIGNALLING JAGUAHR THERAPEUTICS PTE LTD (SG) 2025-04-24 US disclosed
US-20250122205-A1 INDOLE AHR INHIBITORS AND USES THEREOF PAHR THERAPEUTICS, INC. 2025-04-17 US disclosed
US-12077542-B2 Indole AHR inhibitors and uses thereof Ikena Oncology, Inc. (US) 2024-09-03 US disclosed
EP-4396191-A1 COMPOUNDS USEFUL IN MODULATION OF AHR SIGNALLING JAGUAHR THERAPEUTICS PTE LTD (SG) 2024-07-10 EP disclosed
CN-118076613-A Compounds useful for modulating AhR signaling 捷豹治疗有限公司 2024-05-24 CN disclosed
CN-117586428-A Biomass-based macromolecular ultraviolet absorber and preparation method and application thereof 浙江沛格科技有限公司 2024-02-23 CN disclosed
US-4827032-A INTERMEDIATES FOR ANTICOAGULANTS BAYER AKTIENGESELLSCHAFT (DE) 1989-05-02 US disclosed
EP-0242518-A1 Cycloalkano[1,2-b]indole-sulfonamides BAYER AG (DE) 1987-10-28 EP disclosed
CN-87100773-A Cycloalkanes is [1,2-b] indoles-sulfamide compound also 1987-09-02 CN disclosed
US-4257952-A PSYCHOTROPIC DRUGS, ANALGESICS, ANTIHISTAMINES STERLING DRUG INC. (US) 1981-03-24 US disclosed
US-4257952-A PSYCHOTROPIC DRUGS, ANALGESICS, ANTIHISTAMINES STERLING DRUG INC. (US) 1981-03-24 US disclosed
US-4172834-A ANALGESICS, ANTIHISTAMINES AND PSYCHOTROPIC AGENTS STERLING DRUG INC. (US) 1979-10-30 US disclosed
US-4172834-A ANALGESICS, ANTIHISTAMINES AND PSYCHOTROPIC AGENTS STERLING DRUG INC. (US) 1979-10-30 US disclosed
US-4062864-A ANALGESIC, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1977-12-13 US disclosed
US-3959309-A ANALGESICS, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1976-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250129092-A1 COMPOUNDS USEFUL IN MODULATION OF AHR SIGNALLING AHR, ARNT, AIPL1 NR2E1 105/4885HTR6 340/4885HTR1B 693/4885
US-20250122205-A1 INDOLE AHR INHIBITORS AND USES THEREOF AHR, ARNT, IDO1 NR2E1 391/4885HTR6 39/4885HTR1B 76/4885
US-12077542-B2 Indole AHR inhibitors and uses thereof AHR, ARNT, IDO1 NR2E1 391/4885HTR6 39/4885HTR1B 76/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.