SCHEMBL28867414

SCHEMBL28867414

Cc1noc(NS(=O)(=O)c2ccc(S(=O)(=O)N(C)C)cc2)c1C1=CCNCC1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 17/20 0.45
EDNRB P24530 15/20 0.43
HTR6 P50406 1/20 0.42
MEN1 O00255 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
ADRA1A P35348 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29932128 0.92 P2RY1 (0.39) EDNRAEDNRBHTR6MEN1TSHR
SCHEMBL23536374 0.78 EDNRA (0.42) EDNRAEDNRBMEN1CYP2C9TSHR
SCHEMBL23536530 0.74 KIT (0.46) EDNRAEDNRBHTR6
SCHEMBL29932046 0.72 EDNRA (0.41) EDNRAEDNRBMEN1KMT2A
SCHEMBL28867443 0.71 SCN9A (0.38) HTR6
SCHEMBL29948618 0.71 KMT2A (0.38) EDNRAEDNRBMEN1CYP2C9TSHR
SCHEMBL7221292 0.64 EDNRA (0.71) EDNRAEDNRBMEN1CYP2C9TSHR
SCHEMBL29071636 0.63 HTR2C (0.51) HTR6
SCHEMBL7849896 0.63 EDNRA (1.00) EDNRAEDNRBMEN1CYP2C9TSHR
SCHEMBL8479975 0.61 EDNRA (0.66) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115087440-A TRPML modulators 卡斯玛治疗公司 2022-09-20 CN disclosed