SCHEMBL23536374

SCHEMBL23536374

Cc1noc(NS(=O)(=O)c2ccc(S(=O)(=O)N(C)C)cc2)c1C1=CCN(C(=O)O)CC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 14/20 0.42
EDNRB P24530 12/20 0.42
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TSHR P16473 2/20 0.39
TP53 P04637 1/20 0.39
MEN1 O00255 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ADRA1A P35348 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23536530 0.88 KIT (0.46) EDNRAEDNRB
SCHEMBL29948618 0.85 KMT2A (0.38) EDNRAEDNRBHTTNPSR1TSHR
SCHEMBL28867414 0.78 EDNRA (0.45) EDNRAEDNRBTSHRMEN1CYP2C9
SCHEMBL29932046 0.77 EDNRA (0.41) EDNRAEDNRBMEN1KMT2A
Trifluoroacetic Acid SCHEMBL29932128 0.77 P2RY1 (0.39) EDNRAEDNRBHTTTSHRMEN1
SCHEMBL23536239 0.75 ALDH1A1 (0.35) HTTTSHRMEN1CYP2C9CYP2C19
SCHEMBL23536514 0.73 BRD4 (0.40) HTTNPSR1TSHRTP53MEN1
SCHEMBL29071633 0.67 ALDH1A1 (0.46) HTTTSHRTP53MEN1CYP2C19
SCHEMBL18129575 0.65 IGF1R (0.48)
SCHEMBL23536235 0.64 HTR6 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021127337-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed