SCHEMBL29948618

SCHEMBL29948618

CCCCOC(=O)N1CC=C(c2c(C)noc2NS(=O)(=O)c2ccc(S(=O)(=O)N(C)C)cc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
GAA P10253 3/20 0.38
TSHR P16473 3/20 0.38
MAPT P10636 2/20 0.38
HTT P42858 3/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
EDNRA P25101 5/20 0.36
EDNRB P24530 2/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP13 P45452 1/20 0.36
GLA P06280 1/20 0.35
THRB P10828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23536530 0.85 KIT (0.46) EDNRAEDNRB
SCHEMBL23536374 0.85 EDNRA (0.42) KMT2AMEN1TSHRHTTNPSR1
SCHEMBL29948528 0.79 JAK1 (0.37) KMT2AGAAALDH1A1MMP2MMP3
SCHEMBL29948447 0.78 LMNA (0.40) GAATSHRMAPTHTTNPSR1
SCHEMBL28867414 0.71 EDNRA (0.45) KMT2AMEN1TSHRCYP2C9CYP2C19
SCHEMBL29932046 0.71 EDNRA (0.41) KMT2AMEN1MAPTALDH1A1EDNRA
Trifluoroacetic Acid SCHEMBL29932128 0.69 P2RY1 (0.39) KMT2AMEN1TSHRHTTEDNRA
SCHEMBL14144348 0.66 ALDH1A1 (0.54) KMT2AMEN1GAATSHRMAPT
SCHEMBL5460918 0.65 CYP1A2 (0.43) KMT2AMAPTALDH1A1CYP3A4CYP2C9
SCHEMBL29650110 0.64 LMNA (0.47) KMT2AMEN1GAATSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4076423-A1 TRPML MODULATORS Casma Therapeutics, Inc. (US) 2022-10-26 EP disclosed