SCHEMBL28868985

SCHEMBL28868985

CC(C)Oc1cccc(C(=O)c2ccccn2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.57
GRM4 Q14833 3/20 0.50
RAB9A P51151 3/20 0.49
NPC1 O15118 2/20 0.49
PKM P14618 1/20 0.49
CDK5 Q00535 1/20 0.49
CDK5R1 Q15078 1/20 0.49
HSD17B14 Q9BPX1 1/20 0.49
HTT P42858 3/20 0.48
MEN1 O00255 2/20 0.48
GAA P10253 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
LMNA P02545 3/20 0.47
MITF O75030 2/20 0.47
AGTR1 P30556 1/20 0.47
OPRK1 P41145 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
KDM4E B2RXH2 2/20 0.47
ALPL P05186 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968069 1.00 KMT2A (0.57) KMT2AGRM4RAB9ANPC1PKM
SCHEMBL29968072 1.00 KMT2A (0.57) KMT2AGRM4RAB9ANPC1PKM
SCHEMBL7547074 0.85 RAB9A (0.64) KMT2AGRM4RAB9ANPC1PKM
SCHEMBL6322882 0.81 KMT2A (0.61) KMT2ARAB9ANPC1HTTMEN1
SCHEMBL14446354 0.80 ATM (0.59) KMT2ARAB9ANPC1HTTMEN1
SCHEMBL29967930 0.79 PDE4A (0.47) KMT2AGRM4RAB9ANPC1PKM
SCHEMBL29967877 0.79 PDE4A (0.47) KMT2AGRM4RAB9ANPC1PKM
SCHEMBL28337456 0.79 KDM4E (0.69) KMT2AGRM4RAB9ANPC1PKM
SCHEMBL12441772 0.77 KMT2A (0.66) KMT2ARAB9ANPC1PKMHSD17B14
SCHEMBL11798200 0.76 KMT2A (0.64) KMT2ARAB9ANPC1HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109206417-B Opioid receptor agonists and uses thereof 四川海思科制药有限公司 2023-01-03 CN disclosed
CN-115124520-A Opioid receptor agonists and uses thereof 四川海思科制药有限公司 2022-09-30 CN disclosed
CN-109206417-A Opioid receptor agonists and uses thereof 四川海思科制药有限公司 2019-01-15 CN disclosed