SCHEMBL28869838

SCHEMBL28869838

FC(F)(F)c1nc(-c2ccc3ccccc3c2)n(-c2ccccc2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 2/20 0.45
HSD11B1 P28845 2/20 0.45
PTGS1 P23219 1/20 0.43
KMT2A Q03164 3/20 0.42
OPRD1 P41143 1/20 0.42
MAPK9 P45984 2/20 0.42
MAPK10 P53779 2/20 0.42
MAPK8 P45983 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 1/20 0.39
MEN1 O00255 2/20 0.38
GRM1 Q13255 1/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4674384 0.86 PTGS2 (0.42) PDPK1HSD11B1PTGS1KMT2AMAPK9
SCHEMBL28869832 0.85 KMT2A (0.48) PDPK1PTGS1KMT2AMAPK9MAPK10
SCHEMBL28957164 0.84 SMN1; SMN2 (0.54) PTGS1KMT2ASMN1; SMN2CYP1A2NPC1
SCHEMBL4671357 0.84 PDPK1 (0.54) PDPK1PTGS1
SCHEMBL4674149 0.84 PDPK1 (0.69) PDPK1PTGS1LMNA
SCHEMBL28869829 0.81 SMN1; SMN2 (0.44) PTGS1KMT2ASMN1; SMN2MEN1MAPT
SCHEMBL5865649 0.80 PTGS2 (0.60) PTGS1SMN1; SMN2NPC1MAPTRAB9A
SCHEMBL1115174 0.79 HSD11B1 (0.39) PDPK1HSD11B1PTGS1KMT2AOPRD1
SCHEMBL4671346 0.78 HSD11B1 (0.42) PDPK1HSD11B1PTGS1KMT2ASMN1; SMN2
SCHEMBL17011134 0.78 KDM4A (0.43) KMT2AOPRD1MAPK9MAPK10MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093373-A 1, 5-disubstituted-3-fluoroalkyl-1, 2, 4-triazole compound and preparation method and application thereof 江苏省中国科学院植物研究所 2022-09-23 CN disclosed