SCHEMBL28870484

SCHEMBL28870484

COCOc1cccc(C)n1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 1/20 0.43
CCR1 P32246 1/20 0.41
CCR8 P51685 1/20 0.41
HSD17B3 P37058 1/20 0.39
NOS3 P29474 1/20 0.39
NOS2 P35228 1/20 0.39
GRM5 P41594 5/20 0.37
PTPN1 P18031 1/20 0.36
RXRA P19793 3/20 0.35
GRIN1 Q05586 3/20 0.35
GRIN2B Q13224 3/20 0.35
KDM1A O60341 1/20 0.35
HTR7 P34969 2/20 0.35
ASIC3 Q9UHC3 1/20 0.35
P2RX7 Q99572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12092900 0.82 TSHR (0.46) GABRA5CCR1CCR8HSD17B3NOS3
SCHEMBL8234821 0.81 GABRA5 (0.41) GABRA5CCR1CCR8HSD17B3NOS3
SCHEMBL130392 0.79 MAPK8 (0.50) GABRA5CCR1CCR8NOS3NOS2
SCHEMBL29929586 0.78 HTR7 (0.57) GABRA5GRM5PTPN1HTR7
SCHEMBL19436605 0.78 HTR7 (0.57) GABRA5GRM5PTPN1HTR7
SCHEMBL18137723 0.78 GABRA5 (0.44) GABRA5CCR1CCR8HSD17B3NOS3
SCHEMBL15629190 0.78 NOS3 (0.45) GABRA5CCR1CCR8HSD17B3NOS3
SCHEMBL128705 0.76
SCHEMBL29687348 0.76
SCHEMBL12093742 0.76 GRM5 (0.48) GABRA5CCR1CCR8HSD17B3NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105745214-B Tricyclic piperidine compounds 埃科特莱茵药品有限公司 2019-02-19 CN disclosed