SCHEMBL28873146

SCHEMBL28873146

CC(C)(C)OC(=O)NOCCC(O)c1ccc(F)nc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.34
SCN9A Q15858 1/20 0.34
EPHX2 P34913 1/20 0.33
AAK1 Q2M2I8 6/20 0.33
S1PR3 Q99500 1/20 0.33
CA12 O43570 3/20 0.33
CA1 P00915 3/20 0.33
CA2 P00918 3/20 0.33
CA9 Q16790 3/20 0.33
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
P2RY2 P41231 1/20 0.32
TRPA1 O75762 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18921432 0.84 CTSS (0.40)
SCHEMBL18921411 0.83 EPHX2 (0.40) FOLH1EPHX2
SCHEMBL21783498 0.79 ADRB1 (0.34) AAK1CA12CA1CA2CA9
SCHEMBL22232743 0.79 RIPK1 (0.50) CA12CA1
SCHEMBL22456387 0.79 RIPK1 (0.50) CA12CA1
SCHEMBL18921533 0.79 RIPK1 (0.50) CA12CA1
SCHEMBL24454657 0.78 CTSS (0.41) JAK2
SCHEMBL18921453 0.78 CTSS (0.41) JAK2
SCHEMBL29649069 0.78 CTSS (0.41) JAK2
SCHEMBL29641349 0.78 CTSS (0.41) JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602809-B Isoxazolidine derived inhibitors of receptor interacting protein kinase 1(RIPK 1) 戴纳立制药公司 2022-09-30 CN disclosed